SCHEMBL21384576

SCHEMBL21384576

O=C(Nc1ccc(C(F)(F)F)cc1Cl)c1cc(Cl)ccc1NS(=O)(=O)C1CC1

nearest known ligand 0.63

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MRGPRX1 Q96LB2 10/20 0.63
TMPRSS4 Q9NRS4 3/20 0.51
TSPO P30536 1/20 0.47
SMO Q99835 1/20 0.46
PPARG P37231 1/20 0.46
PPARD Q03181 1/20 0.46
NR1H4 Q96RI1 1/20 0.46
IDH1 O75874 1/20 0.46
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
P2RX1 P51575 1/20 0.45
P2RX4 Q99571 1/20 0.45
P2RX7 Q99572 1/20 0.45
CCR9 P51686 1/20 0.44
HRH1 P35367 1/20 0.44
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21394361 0.95 MRGPRX1 (0.58) MRGPRX1TMPRSS4TSPOSMOPPARG
SCHEMBL21394417 0.91 MRGPRX1 (0.53) MRGPRX1TMPRSS4TSPOSMOCA12
SCHEMBL21381353 0.90 MRGPRX1 (0.62) MRGPRX1TMPRSS4TSPOPPARGPPARD
SCHEMBL21394415 0.89 MRGPRX1 (0.61) MRGPRX1TMPRSS4TSPOPPARGPPARD
SCHEMBL21394560 0.89 MRGPRX1 (0.51) MRGPRX1TMPRSS4TSPOSMOCA12
SCHEMBL18341272 0.88 TMPRSS4 (0.54) MRGPRX1TMPRSS4SMOPPARGPPARD
SCHEMBL21384570 0.86 TMPRSS4 (0.55) MRGPRX1TMPRSS4SMOPPARGPPARD
SCHEMBL21394420 0.86 MRGPRX1 (0.56) MRGPRX1TMPRSS4TSPOSMOCA12
SCHEMBL21394554 0.86 MRGPRX1 (0.49) MRGPRX1TMPRSS4TSPOSMOCA12
SCHEMBL24481354 0.85 TMPRSS4 (0.54) MRGPRX1TMPRSS4SMOPPARGPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019179436-A1 ACID AMIDE COMPOUND AND USE THEREOF IN TREATMENT OF CANCERS 成都海创药业有限公司 2019-09-26 WO disclosed
WO-2019179436-A1 ACID AMIDE COMPOUND AND USE THEREOF IN TREATMENT OF CANCERS 成都海创药业有限公司 2019-09-26 WO disclosed