SCHEMBL21394417

SCHEMBL21394417

O=C(Nc1ccc(C(F)(F)F)cc1Cl)c1cc(Br)ccc1NS(=O)(=O)C1CC1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MRGPRX1 Q96LB2 10/20 0.53
TSPO P30536 1/20 0.45
KDM1A O60341 1/20 0.44
SMO Q99835 1/20 0.44
CCKBR P32239 1/20 0.44
SLC10A6 Q3KNW5 2/20 0.44
SLC10A2 Q12908 1/20 0.43
SLC10A1 Q14973 1/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
HRH1 P35367 1/20 0.42
HTT P42858 1/20 0.41
LMNA P02545 1/20 0.41
PKM P14618 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
TMPRSS4 Q9NRS4 1/20 0.41
TRPV1 Q8NER1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21384576 0.91 MRGPRX1 (0.63) MRGPRX1TSPOSMOCA12CA1
SCHEMBL21394554 0.87 MRGPRX1 (0.49) MRGPRX1TSPOSMOCCKBRCA12
SCHEMBL21394560 0.86 MRGPRX1 (0.51) MRGPRX1TSPOSMOCA12CA1
SCHEMBL21394361 0.86 MRGPRX1 (0.58) MRGPRX1TSPOKDM1ASMOCA12
SCHEMBL21394415 0.84 MRGPRX1 (0.61) MRGPRX1TSPOSLC10A6HRH1TMPRSS4
SCHEMBL21394420 0.84 MRGPRX1 (0.56) MRGPRX1TSPOSMOCA12CA1
SCHEMBL21381353 0.81 MRGPRX1 (0.62) MRGPRX1TSPOHRH1LMNATMPRSS4
SCHEMBL21394555 0.81 MRGPRX1 (0.49) MRGPRX1TSPOHRH1TMPRSS4TRPV1
SCHEMBL331420 0.79 TMPRSS4 (0.63) CA12CA1CA2CA9HTT
SCHEMBL30771730 0.79 TMPRSS4 (0.63) CA12CA1CA2CA9HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019179436-A1 ACID AMIDE COMPOUND AND USE THEREOF IN TREATMENT OF CANCERS 成都海创药业有限公司 2019-09-26 WO disclosed