SCHEMBL21394420

SCHEMBL21394420

O=C(Nc1ccc(C(F)(F)F)cc1Cl)c1ccc(F)cc1NS(=O)(=O)C1CC1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MRGPRX1 Q96LB2 10/20 0.56
TSPO P30536 2/20 0.52
HRH1 P35367 1/20 0.48
ALOX15 P16050 5/20 0.47
SMO Q99835 1/20 0.46
TMPRSS4 Q9NRS4 1/20 0.43
TRPV1 Q8NER1 1/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
AVPR2 P30518 1/20 0.42
GPR27 Q9NS67 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21394560 0.88 MRGPRX1 (0.51) MRGPRX1TSPOHRH1SMOTMPRSS4
SCHEMBL21384576 0.86 MRGPRX1 (0.63) MRGPRX1TSPOHRH1SMOTMPRSS4
SCHEMBL21394554 0.85 MRGPRX1 (0.49) MRGPRX1TSPOHRH1SMOTMPRSS4
SCHEMBL21394417 0.84 MRGPRX1 (0.53) MRGPRX1TSPOHRH1SMOTMPRSS4
SCHEMBL21394361 0.82 MRGPRX1 (0.58) MRGPRX1TSPOSMOTMPRSS4CA12
SCHEMBL21394555 0.79 MRGPRX1 (0.49) MRGPRX1TSPOHRH1TMPRSS4TRPV1
SCHEMBL21381353 0.79 MRGPRX1 (0.62) MRGPRX1TSPOHRH1TMPRSS4TRPV1
SCHEMBL21394415 0.76 MRGPRX1 (0.61) MRGPRX1TSPOHRH1TMPRSS4
SCHEMBL20206206 0.76 TMPRSS4 (0.65) ALOX15TMPRSS4TRPV1CA12CA1
SCHEMBL15847536 0.74 MRGPRX1 (0.59) MRGPRX1TSPOHRH1AVPR2GPR27

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019179436-A1 ACID AMIDE COMPOUND AND USE THEREOF IN TREATMENT OF CANCERS 成都海创药业有限公司 2019-09-26 WO disclosed