SCHEMBL21394415

SCHEMBL21394415

O=C(Nc1ccc(C(F)(F)F)cc1Br)c1cc(Cl)ccc1NS(=O)(=O)C1CC1

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MRGPRX1 Q96LB2 11/20 0.61
TMPRSS4 Q9NRS4 4/20 0.49
TSPO P30536 1/20 0.46
PPARG P37231 1/20 0.45
PPARD Q03181 1/20 0.45
NR1H4 Q96RI1 1/20 0.45
P2RX1 P51575 1/20 0.43
P2RX4 Q99571 1/20 0.43
P2RX7 Q99572 1/20 0.43
CCR9 P51686 1/20 0.43
HRH1 P35367 1/20 0.43
SLC10A6 Q3KNW5 1/20 0.42
SLC20A2 Q08357 1/20 0.42
SLC20A1 Q8WUM9 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21384576 0.89 MRGPRX1 (0.63) MRGPRX1TMPRSS4TSPOPPARGPPARD
SCHEMBL21381353 0.88 MRGPRX1 (0.62) MRGPRX1TMPRSS4TSPOPPARGPPARD
SCHEMBL21394555 0.88 MRGPRX1 (0.49) MRGPRX1TMPRSS4TSPOHRH1
SCHEMBL21394361 0.84 MRGPRX1 (0.58) MRGPRX1TMPRSS4TSPOPPARGPPARD
SCHEMBL21394417 0.84 MRGPRX1 (0.53) MRGPRX1TMPRSS4TSPOHRH1SLC10A6
SCHEMBL21394554 0.82 MRGPRX1 (0.49) MRGPRX1TMPRSS4TSPOHRH1
SCHEMBL18341191 0.80 TMPRSS4 (0.75) TMPRSS4P2RX1P2RX4P2RX7
SCHEMBL21384613 0.79 MRGPRX1 (0.61) MRGPRX1TMPRSS4TSPOHRH1
SCHEMBL21394560 0.78 MRGPRX1 (0.51) MRGPRX1TMPRSS4TSPOHRH1
SCHEMBL21384571 0.78 MRGPRX1 (0.60) MRGPRX1TMPRSS4TSPOHRH1SLC10A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019179436-A1 ACID AMIDE COMPOUND AND USE THEREOF IN TREATMENT OF CANCERS 成都海创药业有限公司 2019-09-26 WO disclosed