SCHEMBL21384579

SCHEMBL21384579

COC(=O)c1cc(Cl)cc(C)c1NS(=O)(=O)C1CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX1 Q96LB2 3/20 0.41
FFAR4 Q5NUL3 1/20 0.41
SLC6A3 Q01959 2/20 0.40
ABL1 P00519 1/20 0.39
SCN5A Q14524 1/20 0.39
SCN9A Q15858 1/20 0.39
CTPS1 P17812 2/20 0.38
MAPT P10636 2/20 0.38
ACLY P53396 1/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MAPK1 P28482 1/20 0.38
AURKA O14965 1/20 0.37
TPX2 Q9ULW0 1/20 0.37
ALDH1A1 P00352 2/20 0.36
USP2 O75604 1/20 0.36
SERPINH1 P50454 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21384561 0.86 ACLY (0.48) MRGPRX1FFAR4SCN5ASCN9ACTPS1
SCHEMBL21381359 0.85 MRGPRX1 (0.43) MRGPRX1SLC6A3ABL1SCN5ASCN9A
SCHEMBL21394567 0.84 MRGPRX1 (0.44) MRGPRX1SLC6A3ABL1CTPS1MAPT
SCHEMBL2738023 0.83 KDM4E (0.46) FFAR4SLC6A3ABL1MAPTACLY
SCHEMBL21384614 0.80 MRGPRX1 (0.57) MRGPRX1SLC6A3ABL1ACLY
SCHEMBL11561114 0.77 FFAR4 (0.40) FFAR4SLC6A3ABL1MAPTACLY
SCHEMBL2657833 0.74 ABL1 (0.47) SLC6A3ABL1MAPTMEN1LMNA
SCHEMBL21384541 0.72 ABL1 (0.48) MRGPRX1SLC6A3ABL1MAPTACLY
SCHEMBL17803504 0.71 ABL1 (0.39) MRGPRX1ABL1CTPS1ACLYMEN1
SCHEMBL21384566 0.71 MRGPRX1 (0.42) MRGPRX1SCN5ASCN9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019179436-A1 ACID AMIDE COMPOUND AND USE THEREOF IN TREATMENT OF CANCERS 成都海创药业有限公司 2019-09-26 WO disclosed
WO-2019179436-A1 ACID AMIDE COMPOUND AND USE THEREOF IN TREATMENT OF CANCERS 成都海创药业有限公司 2019-09-26 WO disclosed