SCHEMBL21384596

SCHEMBL21384596

O=S(=O)(OC1=Cc2cccc(Br)c2CC1)C(F)(F)F

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 7/20 0.34
DRD3 P35462 7/20 0.34
DRD4 P21917 5/20 0.34
HTR1D P28221 2/20 0.32
HTR5A P47898 1/20 0.32
DRD1 P21728 3/20 0.31
DRD5 P21918 3/20 0.31
ABHD6 Q9BV23 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22568962 0.83 DRD2 (0.38) DRD2DRD3DRD4HTR1DHTR5A
SCHEMBL29398439 0.82 DRD2 (0.41) DRD2DRD3DRD4HTR1DHTR5A
SCHEMBL22557831 0.82 DRD2 (0.41) DRD2DRD3DRD4HTR1DHTR5A
SCHEMBL225622 0.77 GPR84 (0.35) DRD2DRD3HTR1D
SCHEMBL30152331 0.77 GPR84 (0.35) DRD2DRD3HTR1D
SCHEMBL22557845 0.75 DRD2 (0.39) DRD2DRD3DRD4HTR1DHTR5A
SCHEMBL19230505 0.72 SRD5A1 (0.33) DRD2DRD3HTR1DABHD6
SCHEMBL29399362 0.69 DRD2 (0.43) DRD2DRD3DRD4HTR1DHTR5A
SCHEMBL22569050 0.69 DRD2 (0.43) DRD2DRD3DRD4HTR1DHTR5A
SCHEMBL4306683 0.69 MAOA (0.38) DRD2DRD3DRD4HTR1DDRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111630043-B Compound containing ring, preparation method and application thereof in medicine 四川科伦博泰生物医药股份有限公司 2022-02-15 CN disclosed
CN-111630043-A Compound containing ring, preparation method and application thereof in medicine 四川科伦博泰生物医药股份有限公司 2020-09-04 CN disclosed
WO-2019179369-A1 RING-CONTAINING COMPOUND, PREPARATION METHOD THEREFOR, AND MEDICAL APPLICATION THEREOF 四川科伦博泰生物医药股份有限公司 2019-09-26 WO disclosed