SCHEMBL21385115

SCHEMBL21385115

CCOc1ccn(-c2ccc(C(F)(F)F)cc2)c(=O)c1C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
MCHR1 Q99705 1/20 0.41
MET P08581 5/20 0.41
AXL P30530 2/20 0.41
MST1R Q04912 4/20 0.40
PLK4 O00444 1/20 0.40
ABL1 P00519 1/20 0.40
NTRK1 P04629 1/20 0.40
LCK P06239 1/20 0.40
RET P07949 1/20 0.40
KIT P10721 1/20 0.40
PDGFRA P16234 1/20 0.40
PRKACA P17612 1/20 0.40
KDR P35968 1/20 0.40
FLT3 P36888 1/20 0.40
ABL2 P42684 1/20 0.40
FRK P42685 1/20 0.40
TYRO3 Q06418 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL721541 0.87 MET (0.50) METAXLMST1RPLK4ABL1
SCHEMBL16366161 0.86 LMNA (0.41) METAXLMST1RPLK4ABL1
SCHEMBL15506038 0.85 GLA (0.43) METAXLMST1RPLK4ABL1
SCHEMBL21383502 0.85 MET (0.43) METAXLMST1RPLK4ABL1
SCHEMBL21385290 0.84 MEN1 (0.45) MET
SCHEMBL22234532 0.80 MET (0.43) METAXLMST1RPLK4ABL1
SCHEMBL21383448 0.78 AXL (0.43) METAXLMST1RPLK4ABL1
SCHEMBL18186587 0.77 MET (0.53) METAXLMST1RPLK4ABL1
SCHEMBL14705756 0.77 MET (0.50) METAXLMST1RPLK4ABL1
SCHEMBL23071634 0.76 MET (0.52) METAXLMST1RPLK4ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3762392-B1 THIENOPYRIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING SAME WELLMARKER BIO CO LTD (KR) 2024-05-15 EP disclosed
US-11447500-B2 Thienopyridine derivatives and pharmaceutical composition comprising same WELLMARKER BIO CO., LTD. (KR) 2022-09-20 US disclosed
US-20220288043-A1 THIENOPYRIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING SAME WELLMARKER BIO CO, LTD. (KR) 2022-09-15 US disclosed
CN-111295386-B Thienopyridine derivatives and pharmaceutical compositions containing the same 伟迈可生物有限公司 2022-09-06 CN disclosed
US-20210317133-A1 THIENOPYRIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING SAME WELLMARKER BIO CO., LTD. (KR) 2021-10-14 US disclosed
US-20210317133-A1 THIENOPYRIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING SAME WELLMARKER BIO CO., LTD. (KR) 2021-10-14 US disclosed
EP-3762392-A1 THIENOPYRIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING SAME Wellmarker Bio Co., Ltd. (KR) 2021-01-13 EP disclosed
CN-111295386-A Thienopyridine derivatives and pharmaceutical compositions containing the same 伟迈可生物有限公司 2020-06-16 CN disclosed
WO-2019182274-A1 THIENOPYRIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING SAME WELLMARKER BIO CO., LTD. (KR) 2019-09-26 WO disclosed
WO-2019182274-A1 THIENOPYRIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING SAME WELLMARKER BIO CO., LTD. (KR) 2019-09-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11447500-B2 Thienopyridine derivatives and pharmaceutical composition comprising same MAP4K5, MAP4K2, MAP3K9 CYP1A2 1373/4885CYP2C9 868/4885CYP2C19 563/4885
US-20210317133-A1 THIENOPYRIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING SAME MAP4K5, MAP4K2, MAP3K9 CYP1A2 1373/4885CYP2C9 868/4885CYP2C19 563/4885
US-20220288043-A1 THIENOPYRIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING SAME PRKACA, MAP4K5, MAPKAPK5 CYP1A2 2343/4885CYP2C9 1532/4885CYP2C19 1040/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.