SCHEMBL21386552

SCHEMBL21386552

Cc1ccc(C#Cc2ccc(-c3ccc(N=C=S)c(C)c3)cc2F)cc1

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.34
CYP11B2 P19099 2/20 0.34
AAK1 Q2M2I8 1/20 0.30
AR P10275 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21386561 0.94 CYP11B1 (0.33) CYP11B1CYP11B2AR
SCHEMBL21386531 0.94 FFAR1 (0.30) CYP11B1CYP11B2
SCHEMBL17506887 0.88 CYP11B1 (0.34) CYP11B1CYP11B2AAK1AR
SCHEMBL29305748 0.87 GRM5 (0.35) AAK1
SCHEMBL19057530 0.85 CYP11B1 (0.35) CYP11B1CYP11B2AAK1AR
SCHEMBL29305752 0.85 FFAR1 (0.32)
SCHEMBL21386559 0.81 GRM5 (0.35) AAK1
SCHEMBL22622863 0.81 NAAA (0.33)
SCHEMBL12011040 0.81 CYP11B1 (0.43) CYP11B1CYP11B2AAK1AR
SCHEMBL29305779 0.80 CYP3A4 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240072425-A1 AROMATIC ISOTHIOCYANATES MERCK PATENT GMBH (DE) 2024-02-29 US disclosed
US-11834599-B2 Aromatic isothiocyanates MERCK PATENT GMBH (DE) 2023-12-05 US disclosed
US-11739265-B2 Aromatic isothiocyanates MERCK PATENT GMBH (DE) 2023-08-29 US disclosed
EP-3739020-B1 LIQUID-CRYSTALLINE MEDIUM MERCK PATENT GMBH (DE) 2023-08-23 EP disclosed
WO-2022129018-A1 HETEROAROMATIC ISOTHIOCYANATES MERCK PATENT GMBH (DE) 2022-06-23 WO disclosed
WO-2022128845-A1 HETEROAROMATIC ISOTHIOCYANATES MERCK PATENT GMBH (DE) 2022-06-23 WO disclosed
US-11306251-B2 Liquid-crystalline medium MERCK PATENT GMBH (DE) 2022-04-19 US disclosed
US-11268026-B2 Liquid-crystalline medium MERCK PATENT GMBH (DE) 2022-03-08 US disclosed
WO-2022043376-A1 AROMATIC ISOTHIOCYANATES MERCK PATENT GMBH (DE) 2022-03-03 WO disclosed
WO-2021116080-A1 AROMATIC ISOTHIOCYANATES MERCK PATENT GMBH (DE) 2021-06-17 WO disclosed
EP-3739020-A1 LIQUID-CRYSTALLINE MEDIUM Merck Patent GmbH (DE) 2020-11-18 EP disclosed
US-20200347301-A1 Isothiocyanato-tolanes MERCK PATENT GMBH (DE) 2020-11-05 US disclosed
EP-3733816-A1 ISOTHIOCYANATO-TOLANES Merck Patent GmbH (DE) 2020-11-04 EP disclosed
EP-3543313-B1 LIQUID-CRYSTALLINE MEDIUM MERCK PATENT GMBH (DE) 2020-10-07 EP disclosed
EP-3543314-B1 LIQUID-CRYSTALLINE MEDIUM MERCK PATENT GMBH (DE) 2020-09-09 EP disclosed
US-20190352564-A1 LIQUID-CRYSTALLINE MEDIUM MERCK PATENT GMBH (DE) 2019-11-21 US disclosed
US-20190292458-A1 LIQUID-CRYSTALLINE MEDIUM MERCK PATENT GMBH (DE) 2019-09-26 US disclosed
US-20190292460-A1 LIQUID-CRYSTALLINE MEDIUM MERCK PATENT GMBH (DE) 2019-09-26 US disclosed
EP-3543314-A1 LIQUID-CRYSTALLINE MEDIUM Merck Patent GmbH (DE) 2019-09-25 EP disclosed
EP-3543313-A1 LIQUID-CRYSTALLINE MEDIUM Merck Patent GmbH (DE) 2019-09-25 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240072425-A1 AROMATIC ISOTHIOCYANATES TRPA1, TRPC1, CRY1 CYP11B1 4276/4885CYP11B2 4408/4885AAK1 235/4885
US-11739265-B2 Aromatic isothiocyanates TRPA1, CRY1, FOXM1 CYP11B1 4339/4885CYP11B2 4429/4885AAK1 258/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.