SCHEMBL21386735

SCHEMBL21386735

C=CC(=O)N1CCC[C@@H](Nc2ncnc(N)c2C(=N)c2ccc(Oc3ccccc3)cn2)C1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 16/20 0.76
EGFR P00533 5/20 0.69
JAK3 P52333 5/20 0.51
JAK1 P23458 1/20 0.51
TEC P42680 4/20 0.50
BMX P51813 3/20 0.50
LYN P07948 3/20 0.50
TXK P42681 2/20 0.50
RIPK2 O43353 2/20 0.50
LCK P06239 2/20 0.50
FYN P06241 2/20 0.50
YES1 P07947 2/20 0.50
HCK P08631 2/20 0.50
SRC P12931 2/20 0.50
CSK P41240 2/20 0.50
PTK6 Q13882 2/20 0.50
FGFR2 P21802 2/20 0.50
ITK Q08881 2/20 0.50
NR1I2 O75469 1/20 0.50
SLC22A3 O75751 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18877721 0.91 BTK (0.86) BTKEGFRJAK3JAK1TEC
SCHEMBL14228143 0.91 BTK (0.86) BTKEGFRJAK3JAK1TEC
SCHEMBL21386748 0.87 BTK (0.74) BTKEGFRJAK3JAK1TEC
SCHEMBL19533419 0.86 BTK (1.00) BTKEGFRJAK3JAK1TEC
SCHEMBL19533436 0.86 BTK (1.00) BTKEGFRJAK3JAK1TEC
SCHEMBL17816357 0.86 BTK (0.77) BTKEGFRTECBMXITK
SCHEMBL21386777 0.85 BTK (0.75) BTKEGFRJAK3JAK1BLK
SCHEMBL21386710 0.83 BTK (0.68) BTKEGFRJAK3JAK1ITK
SCHEMBL21386778 0.83 BTK (0.66) BTKEGFRJAK3JAK1ITK
SCHEMBL21386723 0.83 BTK (0.68) BTKEGFRJAK3BMXHCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3543239-A1 SELECTIVE BRUTON'S TYROSINE KINASE INHIBITOR AND USE THEREOF Hangzhou Hertz Pharmaceutical Co., Ltd. (CN) 2019-09-25 EP disclosed