SCHEMBL21386782

SCHEMBL21386782

C=CC(=O)N1CC[C@@H](Nc2ncnc(N)c2C(=N)c2ccc(Oc3ccccc3)nc2)C1

nearest known ligand 0.67

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BTK Q06187 20/20 0.67
EGFR P00533 2/20 0.57
KCNH2 Q12809 2/20 0.48
TEC P42680 1/20 0.48
BMX P51813 1/20 0.48
CD69 Q07108 1/20 0.48
ITK Q08881 1/20 0.48
ERBB4 Q15303 1/20 0.48
GP6 Q9HCN6 1/20 0.48
NUDT5 Q9UKK9 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21386777 0.95 BTK (0.75) BTKEGFR
SCHEMBL17816357 0.91 BTK (0.77) BTKEGFRKCNH2TECBMX
SCHEMBL21386770 0.88 BTK (0.66) BTKEGFRITK
SCHEMBL21386780 0.88 BTK (0.66) BTKEGFRITK
SCHEMBL21386692 0.88 BTK (0.54) BTKEGFRTECBMXITK
SCHEMBL21386739 0.87 BTK (0.54) BTKEGFRITK
SCHEMBL21386733 0.87 BTK (0.62) BTKEGFRKCNH2ITK
SCHEMBL18877721 0.86 BTK (0.86) BTKEGFRKCNH2TECBMX
SCHEMBL14228143 0.86 BTK (0.86) BTKEGFRKCNH2TECBMX
SCHEMBL21386748 0.86 BTK (0.74) BTKEGFRKCNH2TECBMX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3543239-A1 SELECTIVE BRUTON'S TYROSINE KINASE INHIBITOR AND USE THEREOF Hangzhou Hertz Pharmaceutical Co., Ltd. (CN) 2019-09-25 EP disclosed