SCHEMBL2138785

SCHEMBL2138785

COc1cc2c(cc1OC)Cc1cc(OC)c(OC)cc1C2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 1.00
MAPT P10636 2/20 1.00
DRD1 P21728 2/20 0.53
DRD4 P21917 2/20 0.53
DRD5 P21918 2/20 0.53
GAA P10253 2/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
DRD2 P14416 1/20 0.47
DRD3 P35462 1/20 0.47
KDM4E B2RXH2 5/20 0.46
MAOA P21397 5/20 0.46
CHRNA7 P36544 2/20 0.46
MAOB P27338 2/20 0.46
SLC6A4 P31645 1/20 0.46
ALDH1A1 P00352 4/20 0.43
GLA P06280 2/20 0.43
ACHE P22303 1/20 0.43
BRD4 O60885 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4571013 1.00 CYP3A4 (1.00) CYP3A4MAPTDRD1DRD4DRD5
SCHEMBL29394312 1.00 CYP3A4 (1.00) CYP3A4MAPTDRD1DRD4DRD5
SCHEMBL22953335 1.00 CYP3A4 (1.00) CYP3A4MAPTDRD1DRD4DRD5
SCHEMBL13456132 0.92 MAPT (0.84) CYP3A4MAPTDRD1DRD4DRD5
SCHEMBL6904036 0.92 MAPT (0.84) CYP3A4MAPTDRD1DRD4DRD5
SCHEMBL25591699 0.88 CYP3A4 (0.78) CYP3A4MAPTDRD1DRD4DRD5
SCHEMBL29460958 0.88 CYP3A4 (0.78) CYP3A4MAPTDRD1DRD4DRD5
SCHEMBL13508341 0.87 MAPT (0.76) CYP3A4MAPTDRD1DRD4DRD5
SCHEMBL7981630 0.86 MAPT (0.75) CYP3A4MAPTDRD1DRD4DRD5
SCHEMBL12595457 0.84 MAPT (0.71) CYP3A4MAPTDRD1DRD4DRD5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7862775-B2 Determination of explosives including RDX MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2011-01-04 US disclosed
US-7862775-B2 Determination of explosives including RDX MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2011-01-04 US disclosed
US-20100303672-A1 DETERMINATION OF EXPLOSIVES INCLUDNIG RDX MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2010-12-02 US disclosed
US-7666684-B2 luminescence emission MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2010-02-23 US disclosed
US-20100022011-A1 DETERMINATION OF EXPLOSIVES INCLUDING RDX MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2010-01-28 US disclosed
WO-2008130376-A2 DETERMINATION OF EXPLOSIVES INCLUDING RDX MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2008-10-30 WO disclosed
WO-2008130376-A2 DETERMINATION OF EXPLOSIVES INCLUDING RDX MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2008-10-30 WO disclosed