SCHEMBL21390826

SCHEMBL21390826

COc1cc(F)c2nc(CCCC(=O)CC(C)(C)C)n(C3CCC3)c2c1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 1/20 0.35
BRD4 O60885 9/20 0.34
CREBBP Q92793 9/20 0.34
MAPK1 P28482 1/20 0.33
ACACB O00763 1/20 0.32
CDK4 P11802 1/20 0.32
CCND1 P24385 1/20 0.32
CCND3 P30281 1/20 0.32
CDK6 Q00534 1/20 0.32
HDAC1 Q13547 2/20 0.32
IDH1 O75874 1/20 0.32
PKM P14618 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
ALDH1A1 P00352 1/20 0.31
TBXA2R P21731 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21390672 0.90 BRD4 (0.34) BRD4CREBBPACACBCDK4CCND1
SCHEMBL23132029 0.84 HDAC1 (0.33) BRD4CREBBPCDK4CCND1CCND3
SCHEMBL21391103 0.84 HDAC1 (0.33) BRD4CREBBPCDK4CCND1CCND3
SCHEMBL21390898 0.84 HDAC1 (0.32) CDK4CCND1CCND3CDK6HDAC1
SCHEMBL21390933 0.83 CDK4 (0.32) CDK4CCND1CCND3CDK6HDAC1
SCHEMBL21390697 0.83 BRD4 (0.33) BRD4CREBBPACACBCDK4CCND1
SCHEMBL21390935 0.82 HDAC1 (0.33) BRD4CREBBPCDK4CCND1CCND3
SCHEMBL21391027 0.80 CDK4 (0.32) CDK4CCND1CCND3CDK6HDAC1
SCHEMBL21390822 0.79 CYP19A1 (0.33) CDK4CCND1CCND3CDK6HDAC1
SCHEMBL21354610 0.78 CACNA1H (0.40) CACNA1HBRD4CREBBPMAPK1ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019183148-A1 KV7 CHANNEL ACTIVATORS COMPOSITIONS AND METHODS OF USE KNOPP BIOSCIENCES LLC (US) 2019-09-26 WO disclosed