SCHEMBL21390914

SCHEMBL21390914

CC1(n2c(CCCC(=O)CC3CC(F)(F)C3(F)F)nc3cc(F)ccc32)CCC1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 2/20 0.35
AGTR2 P50052 2/20 0.35
TBXA2R P21731 6/20 0.33
IDH1 O75874 2/20 0.33
HDAC3 O15379 1/20 0.33
PTGS1 P23219 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC10 Q969S8 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
HDAC5 Q9UQL6 1/20 0.33
CYP11B1 P15538 1/20 0.30
CYP11B2 P19099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21391090 0.97 AGTR1 (0.35) AGTR1AGTR2TBXA2RIDH1HDAC3
SCHEMBL21390871 0.83
SCHEMBL21390862 0.79 AGTR1 (0.37) AGTR1AGTR2TBXA2RIDH1HDAC3
SCHEMBL21354576 0.79 IDH1 (0.35) IDH1
SCHEMBL21390717 0.76 ACACB (0.31)
SCHEMBL21390703 0.73
SCHEMBL23329655 0.72 TBXA2R (0.33) TBXA2R
SCHEMBL21391115 0.72
SCHEMBL26008187 0.72 IDH1 (0.35) IDH1
SCHEMBL21391084 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019183148-A1 KV7 CHANNEL ACTIVATORS COMPOSITIONS AND METHODS OF USE KNOPP BIOSCIENCES LLC (US) 2019-09-26 WO disclosed