SCHEMBL21392957

SCHEMBL21392957

Nc1ncnc2c1ncn2[C@H]1CC[C@@H](CNS(=O)(=O)O)O1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BLM P54132 3/20 0.55
NFKB1 P19838 2/20 0.55
CYP3A4 P08684 2/20 0.55
CYP1A2 P05177 1/20 0.55
THPO P40225 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
ADA P00813 1/20 0.50
MAPK1 P28482 3/20 0.49
ALDH1A1 P00352 2/20 0.49
PI4KA P42356 2/20 0.49
PI4K2B Q8TCG2 2/20 0.49
PI4K2A Q9BTU6 2/20 0.49
PI4KB Q9UBF8 2/20 0.49
TP53 P04637 1/20 0.49
CYP2C9 P11712 1/20 0.49
HSD17B10 Q99714 1/20 0.49
MEN1 O00255 1/20 0.49
APEX1 P27695 1/20 0.49
KMT2A Q03164 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21637076 0.89 ADA (0.48) BLMNFKB1CYP3A4CYP1A2THPO
SCHEMBL21637027 0.87 ALDH1A1 (0.44) BLMNFKB1CYP3A4CYP1A2THPO
SCHEMBL21636983 0.85 NFKB1 (0.47) BLMNFKB1CYP3A4CYP1A2THPO
SCHEMBL19941795 0.84 ADA (0.51) BLMNFKB1CYP3A4CYP1A2THPO
SCHEMBL21636996 0.82 ALDH1A1 (0.71) CYP1A2MAPK1ALDH1A1LMNAALB
SCHEMBL10381269 0.82 ADA (0.65) BLMNFKB1SMN1; SMN2ADAMAPK1
SCHEMBL1374909 0.82 ADA (0.65) BLMNFKB1SMN1; SMN2ADAMAPK1
SCHEMBL3541 0.82 ADA (0.65) BLMNFKB1SMN1; SMN2ADAMAPK1
SCHEMBL20419221 0.82 ADA (0.65) BLMNFKB1SMN1; SMN2ADAMAPK1
SCHEMBL9197787 0.82 ADA (0.65) BLMNFKB1SMN1; SMN2ADAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020016782-A1 CYCLIC DINUCLEOTIDES AS STING AGONISTS JANSSEN BIOTECH, INC. (US) 2020-01-23 WO disclosed
WO-2019180683-A1 STING MODULATOR COMPOUNDS WITH SULFAMATE LINKAGES, AND METHODS OF MAKING AND USING TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2019-09-26 WO disclosed