SCHEMBL21393521

SCHEMBL21393521

Nc1cc(F)cc(C(F)F)c1

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
KCNH2 Q12809 1/20 0.33
IDO1 P14902 1/20 0.31
TDO2 P48775 1/20 0.31
FFAR4 Q5NUL3 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13401017 0.84 CYP3A4 (0.33)
SCHEMBL27874501 0.78 CA12 (0.38) CES2CES1IDO1TDO2
SCHEMBL13491971 0.78 ALDH1A1 (0.39) CES2CES1IDO1TDO2
SCHEMBL25078128 0.76 IDO1 (0.33) CES2CES1IDO1TDO2
Hydrochloric Acid SCHEMBL30496913 0.75 IDO1 (0.36) CES2CES1IDO1TDO2
Hydrochloric Acid SCHEMBL29109435 0.75 IDO1 (0.36) CES2CES1IDO1TDO2
Hydrochloric Acid SCHEMBL29109434 0.75 IDO1 (0.36) CES2CES1IDO1TDO2
SCHEMBL1100115 0.74
SCHEMBL69602 0.74
SCHEMBL11803395 0.73 CYP3A4 (0.55) KCNH2IDO1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11078168-B2 Substituted N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase Phenex Discovery Verwaltungs-GmbH (DE) 2021-08-03 US disclosed
US-20190292160-A1 SUBSTITUTED N-HYDROXYAMIDINOHETEROCYCLES AS MODULATORS OF INDOLEAMINE 2,3-DIOXYGENASE Phenex Discovery Verwaltungs-GmbH (DE) 2019-09-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11078168-B2 Substituted N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase IDO1, IDO2, INMT CES2 2784/4885CES1 794/4885KCNH2 3927/4885
US-20190292160-A1 SUBSTITUTED N-HYDROXYAMIDINOHETEROCYCLES AS MODULATORS OF INDOLEAMINE 2,3-DIOXYGENASE IDO1, IDO2, INMT CES2 2784/4885CES1 794/4885KCNH2 3927/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.