SCHEMBL21393634

SCHEMBL21393634

Bc1cncc(F)c1C(=O)OC

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.40
CYP11B2 P19099 1/20 0.39
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37
CA14 Q9ULX7 1/20 0.37
ALDH1A1 P00352 3/20 0.36
TSHR P16473 3/20 0.35
POLB P06746 1/20 0.35
KDM4E B2RXH2 2/20 0.34
GLA P06280 1/20 0.34
GAA P10253 1/20 0.34
LMNA P02545 1/20 0.34
NPSR1 Q6W5P4 1/20 0.33
MAPK1 P28482 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ALPL P05186 2/20 0.33
CYP3A4 P08684 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3348369 0.87 ATM (0.46) ATMCYP11B2CA12CA1CA2
SCHEMBL20187531 0.84 ATM (0.44) ATMCYP11B2CA12CA1CA2
SCHEMBL13067195 0.81 CYP2C9 (0.44) CA12CA1CA2CA7CA9
SCHEMBL6921530 0.79 CYP11B2 (0.35) CYP11B2CYP3A4HPGD
SCHEMBL25190713 0.79 ALDH1A1 (0.49) ATMCYP11B2CA12CA1CA2
SCHEMBL17197218 0.79 CYP11B2 (0.41) ATMCYP11B2CA12CA1CA2
SCHEMBL20187445 0.79 ATM (0.43) ATMCYP11B2CA12CA1CA2
SCHEMBL14392455 0.77 HCAR2 (0.39) ALDH1A1POLBKDM4ELMNA
SCHEMBL22620862 0.76 CYP11B2 (0.40) ATMCYP11B2CA12CA1CA2
SCHEMBL24746934 0.75 L3MBTL1 (0.37) ATMCYP11B2CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019182925-A1 OXADIAZOLE TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS GENENTECH, INC. (US) 2019-09-26 WO disclosed