SCHEMBL21393782

SCHEMBL21393782

CC(=O)c1c(C)ccnc1/N=C\C(C)C(C)C

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.32
CYP2C19 P33261 1/20 0.32
PLAU P00749 1/20 0.30
ALDH1A1 P00352 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21393825 0.73 CSNK1A1 (0.33) CYP2C19PLAUALDH1A1
SCHEMBL31662998 0.67 CSNK1A1 (0.38) CYP2C19ALDH1A1
SCHEMBL6628045 0.67 CSNK1A1 (0.38) CYP2C19ALDH1A1
SCHEMBL25932246 0.64 CSNK1A1 (0.36) CYP2C19ALDH1A1
SCHEMBL28700162 0.64 NAPRT (0.37) CYP2C19ALDH1A1
SCHEMBL17692459 0.64 SMN1; SMN2 (0.37) CYP2C19ALDH1A1
SCHEMBL21393794 0.61 KDM4E (0.34) CYP1A2CYP2C19ALDH1A1
SCHEMBL696352 0.60 THRB (0.56) CYP1A2ALDH1A1
SCHEMBL6578250 0.60 KDM4E (0.43) CYP1A2ALDH1A1
SCHEMBL12824158 0.59 THRB (0.48) CYP1A2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019182925-A1 OXADIAZOLE TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS GENENTECH, INC. (US) 2019-09-26 WO disclosed