SCHEMBL21394824

SCHEMBL21394824

Cn1ccc(C(=O)Nc2ccc(Cc3ccc(F)c(F)c3)cn2)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.47
RAB9A P51151 6/20 0.47
SMN1; SMN2 Q16637 5/20 0.47
TSHR P16473 1/20 0.47
GSK3B P49841 1/20 0.44
DYRK1A Q13627 1/20 0.44
BACE1 P56817 4/20 0.42
BACE2 Q9Y5Z0 2/20 0.42
NFKB1 P19838 2/20 0.41
NFKB2 Q00653 2/20 0.41
RELA Q04206 2/20 0.41
HPGD P15428 1/20 0.41
CACNA1G O43497 4/20 0.41
CACNA1H O95180 4/20 0.41
CACNA1I Q9P0X4 4/20 0.41
LMNA P02545 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
TDP1 Q9NUW8 1/20 0.40
MEN1 O00255 1/20 0.40
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29357599 1.00 NPC1 (0.47) NPC1RAB9ASMN1; SMN2TSHRGSK3B
SCHEMBL29358408 0.88 NPC1 (0.47) NPC1RAB9ASMN1; SMN2TSHRGSK3B
SCHEMBL21394690 0.88 NPC1 (0.47) NPC1RAB9ASMN1; SMN2TSHRGSK3B
SCHEMBL21394575 0.87 RAB9A (0.65) NPC1RAB9ASMN1; SMN2TSHRCACNA1G
SCHEMBL29442886 0.87 RAB9A (0.65) NPC1RAB9ASMN1; SMN2TSHRCACNA1G
SCHEMBL21394867 0.86 NPC1 (0.49) NPC1RAB9ASMN1; SMN2TSHRGSK3B
SCHEMBL29357020 0.86 NPC1 (0.49) NPC1RAB9ASMN1; SMN2TSHRGSK3B
SCHEMBL21394578 0.85 L3MBTL1 (0.46) NPC1RAB9ASMN1; SMN2TSHRCACNA1H
SCHEMBL29355468 0.85 L3MBTL1 (0.46) NPC1RAB9ASMN1; SMN2TSHRCACNA1H
SCHEMBL21395020 0.84 CACNA1H (0.43) NPC1RAB9ASMN1; SMN2TSHRCACNA1G

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118084800-A Compounds and uses thereof 詹森药业有限公司 2024-05-28 CN disclosed
CN-118084801-A Compounds and uses thereof 詹森药业有限公司 2024-05-28 CN disclosed
CN-112312913-B Compounds and uses thereof 詹森药业有限公司 2024-03-08 CN disclosed
CN-114174273-A Compounds and uses thereof 优曼尼蒂治疗公司 2022-03-11 CN disclosed
CN-112312913-A Compounds and uses thereof 优曼尼蒂治疗公司 2021-02-02 CN disclosed
WO-2020198026-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-10-01 WO disclosed
WO-2019183587-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed