SCHEMBL21395020

SCHEMBL21395020

Cn1ccc(C(=O)Nc2ccc(Cc3ccc(F)c(F)c3)cn2)nc1=O

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 6/20 0.43
CACNA1G O43497 4/20 0.43
CACNA1I Q9P0X4 4/20 0.43
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
TSHR P16473 1/20 0.40
AHR P35869 1/20 0.37
GRM5 P41594 3/20 0.36
CYP3A4 P08684 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C9 P11712 2/20 0.36
PPARG P37231 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
NTRK1 P04629 1/20 0.36
KCNH2 Q12809 1/20 0.36
RIPK1 Q13546 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21395084 0.89 AHR (0.39) CACNA1HNPC1RAB9ASMN1; SMN2TSHR
SCHEMBL21394649 0.84 P2RX3 (0.45) CACNA1HCACNA1GCACNA1INPC1RAB9A
SCHEMBL29357599 0.84 NPC1 (0.47) CACNA1HCACNA1GCACNA1INPC1RAB9A
SCHEMBL21394824 0.84 NPC1 (0.47) CACNA1HCACNA1GCACNA1INPC1RAB9A
SCHEMBL21395147 0.82 NPC1 (0.39) CACNA1HCACNA1GCACNA1INPC1RAB9A
SCHEMBL21394575 0.80 RAB9A (0.65) CACNA1HCACNA1GCACNA1INPC1RAB9A
SCHEMBL29442886 0.80 RAB9A (0.65) CACNA1HCACNA1GCACNA1INPC1RAB9A
SCHEMBL21394578 0.80 L3MBTL1 (0.46) CACNA1HNPC1RAB9ASMN1; SMN2TSHR
SCHEMBL29355468 0.80 L3MBTL1 (0.46) CACNA1HNPC1RAB9ASMN1; SMN2TSHR
SCHEMBL21395082 0.80 NPC1 (0.43) NPC1RAB9ASMN1; SMN2GRM5CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020198026-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-10-01 WO disclosed
WO-2019183587-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed