SCHEMBL21395070

SCHEMBL21395070

Cn1nc(C(=O)Nc2ccc(Oc3cc(F)cc(Cl)c3)cn2)ccc1=O

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 8/20 0.49
GRM5 P41594 2/20 0.48
CYP1A2 P05177 4/20 0.47
CYP2C9 P11712 4/20 0.47
L3MBTL1 Q9Y468 1/20 0.46
SLC6A3 Q01959 1/20 0.44
KCNH2 Q12809 1/20 0.43
TSHR P16473 1/20 0.41
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21395157 0.94 CYP3A4 (0.47) CYP3A4GRM5CYP1A2CYP2C9L3MBTL1
SCHEMBL29356824 0.87 L3MBTL1 (0.47) CYP3A4GRM5CYP1A2CYP2C9L3MBTL1
SCHEMBL21394821 0.87 L3MBTL1 (0.47) CYP3A4GRM5CYP1A2CYP2C9L3MBTL1
SCHEMBL29359147 0.87 TSHR (0.47) CYP3A4GRM5CYP1A2CYP2C9L3MBTL1
SCHEMBL21394809 0.87 TSHR (0.47) CYP3A4GRM5CYP1A2CYP2C9L3MBTL1
SCHEMBL29357070 0.86 L3MBTL1 (0.47) GRM5L3MBTL1TSHRHTT
SCHEMBL21394806 0.86 L3MBTL1 (0.47) GRM5L3MBTL1TSHRHTT
SCHEMBL21395074 0.83 CYP3A4 (0.53) CYP3A4GRM5CYP1A2CYP2C9
SCHEMBL21394626 0.80 L3MBTL1 (0.46) GRM5L3MBTL1TSHRHTT
SCHEMBL29357041 0.80 L3MBTL1 (0.46) GRM5L3MBTL1TSHRHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020198026-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-10-01 WO disclosed
WO-2019183587-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed