SCHEMBL29359147

SCHEMBL29359147

Cn1nc(C(=O)Nc2ccc(Oc3cccc(F)c3)cn2)ccc1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.47
ABL1 P00519 1/20 0.45
GCK P35557 1/20 0.44
MEN1 O00255 1/20 0.44
POLB P06746 1/20 0.44
KMT2A Q03164 1/20 0.44
NPC1 O15118 1/20 0.43
ALDH1A1 P00352 1/20 0.43
PKM P14618 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
GRM5 P41594 2/20 0.43
NTRK1 P04629 1/20 0.43
CYP3A4 P08684 2/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2C9 P11712 2/20 0.43
SLC6A3 Q01959 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.42
HRH3 Q9Y5N1 1/20 0.42
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21394809 1.00 TSHR (0.47) TSHRABL1GCKMEN1POLB
SCHEMBL21395157 0.91 CYP3A4 (0.47) TSHRGCKGRM5CYP3A4CYP1A2
SCHEMBL21394806 0.89 L3MBTL1 (0.47) TSHRABL1GCKMEN1KMT2A
SCHEMBL29357070 0.89 L3MBTL1 (0.47) TSHRABL1GCKMEN1KMT2A
SCHEMBL21395070 0.87 CYP3A4 (0.49) TSHRGRM5CYP3A4CYP1A2CYP2C9
SCHEMBL29356824 0.86 L3MBTL1 (0.47) TSHRMEN1KMT2ANPC1RAB9A
SCHEMBL21394821 0.86 L3MBTL1 (0.47) TSHRMEN1KMT2ANPC1RAB9A
SCHEMBL29357283 0.82 GCK (0.52) TSHRABL1GCKMEN1POLB
SCHEMBL21394862 0.82 GCK (0.52) TSHRABL1GCKMEN1POLB
SCHEMBL21394512 0.81 TSHR (0.53) TSHRMEN1POLBKMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118084800-A Compounds and uses thereof 詹森药业有限公司 2024-05-28 CN disclosed
CN-118084801-A Compounds and uses thereof 詹森药业有限公司 2024-05-28 CN disclosed
CN-112312913-B Compounds and uses thereof 詹森药业有限公司 2024-03-08 CN disclosed
CN-114174273-A Compounds and uses thereof 优曼尼蒂治疗公司 2022-03-11 CN disclosed
EP-3941908-A1 COMPOUNDS AND USES THEREOF Yumanity Therapeutics, Inc. (US) 2022-01-26 EP disclosed