SCHEMBL21397329

SCHEMBL21397329

COc1ccc(N2CCC(N)CC2)c(F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.47
DRD2 P14416 1/20 0.44
DRD3 P35462 1/20 0.44
HTR3E A5X5Y0 1/20 0.43
HTR3B O95264 1/20 0.43
HTR3A P46098 1/20 0.43
HTR3D Q70Z44 1/20 0.43
HTR3C Q8WXA8 1/20 0.43
KDM1A O60341 1/20 0.43
LMNA P02545 2/20 0.42
TSHR P16473 2/20 0.42
KDM4E B2RXH2 1/20 0.42
CPS1 P31327 5/20 0.42
SSTR2 P30874 1/20 0.41
GAA P10253 1/20 0.40
MAPK1 P28482 1/20 0.40
KMT2A Q03164 1/20 0.39
KYAT1 Q16773 1/20 0.39
KYAT3 Q6YP21 1/20 0.39
AADAT Q8N5Z0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30815847 1.00 ACACB (0.47) ACACBDRD2DRD3HTR3EHTR3B
SCHEMBL21397269 0.84 ACACB (0.44) ACACBHTR3EHTR3BHTR3AHTR3D
SCHEMBL11906870 0.83 KDM4E (0.47) DRD2DRD3HTR3EHTR3BHTR3A
SCHEMBL8129610 0.82 ALDH1A1 (0.51) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL8138147 0.81 ALDH1A1 (0.50) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL27474183 0.80 GAA (0.42) ACACBGAAKMT2A
SCHEMBL13419247 0.80 SSTR2 (0.43) ACACBLMNATSHRSSTR2GAA
SCHEMBL14922713 0.80 LMNA (0.54) DRD2DRD3HTR3EHTR3BHTR3A
SCHEMBL4539952 0.79 ALDH1A1 (0.45) ACACBLMNAKDM4EGAAMAPK1
SCHEMBL2768723 0.78 HTR3A (0.69) DRD2DRD3HTR3EHTR3BHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112574176-B Heteroaryl compound and application thereof 隆泰申医药科技(南京) 有限公司 2024-03-15 CN disclosed
WO-2021057696-A1 HETEROARYL COMPOUND AND APPLICATION THEREOF 隆泰申医药科技(南京)有限公司 2021-04-01 WO disclosed
CN-112574176-A Heteroaryl compound and application thereof 隆泰申医药科技(南京) 有限公司 2021-03-30 CN disclosed
WO-2019179362-A1 AMIDINE AND GUANIDINE DERIVATIVES, PREPARATION METHOD THEREFOR AND MEDICAL USES THEREOF 四川科伦博泰生物医药股份有限公司 2019-09-26 WO disclosed