SCHEMBL21397500

SCHEMBL21397500

CCCC1(CCC)Cc2c(C)cccc2C1N

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
ADRA1D P25100 1/20 0.35
ADRA1A P35348 1/20 0.35
ADRA1B P35368 1/20 0.35
SLC6A2 P23975 2/20 0.33
SLC6A4 P31645 2/20 0.33
SLC6A3 Q01959 2/20 0.33
HTR2A P28223 2/20 0.33
HTR2C P28335 2/20 0.33
HTR2B P41595 2/20 0.33
AADAT Q8N5Z0 1/20 0.31
KDM1A O60341 3/20 0.31
ALDH1A1 P00352 2/20 0.31
MAOA P21397 2/20 0.31
MAOB P27338 2/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
KIF11 P52732 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22515446 0.87 ADRA2A (0.36) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL21397317 0.81 SLC6A2 (0.34) SLC6A2SLC6A4SLC6A3
SCHEMBL22515384 0.79 KDM1A (0.34) SLC6A4SLC6A3HTR2AHTR2CHTR2B
SCHEMBL21397337 0.76 HTR2A (0.37) ADRA2AADRA2BADRA2CADRA1BSLC6A2
SCHEMBL22515237 0.76 KDM1A (0.32) ADRA2AADRA2BADRA2CKDM1A
SCHEMBL21397653 0.70 HTR2A (0.35) ADRA2AADRA2BADRA2CADRA1BSLC6A2
SCHEMBL24091164 0.70 KMT2A (0.40) AADATKMT2AKIF11
SCHEMBL21397670 0.68 HTR2A (0.33) ADRA2AADRA2BADRA2CADRA1AADRA1B
SCHEMBL21940878 0.67 SLC6A3 (0.38) ADRA2ASLC6A2SLC6A4SLC6A3HTR2B
SCHEMBL21940662 0.67 SLC6A3 (0.38) ADRA2ASLC6A2SLC6A4SLC6A3HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019183367-A1 SHP2 PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF RELAY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed