SCHEMBL21397520

SCHEMBL21397520

CCCC1(CCC(C)C)Cc2ccc(C(=O)N(C)C)cc2C1N

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.38
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
BACE1 P56817 1/20 0.32
OTUD7B Q6GQQ9 1/20 0.31
PDK2 Q15119 1/20 0.30
DPP4 P27487 1/20 0.30
SLC6A2 P23975 2/20 0.30
SLC6A4 P31645 2/20 0.30
SLC6A3 Q01959 2/20 0.30
KDM2B Q8NHM5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21397670 0.76 HTR2A (0.33) DRD2OPRK1
SCHEMBL24388797 0.73 SLC6A2 (0.39) DRD2BACE1OTUD7BPDK2SLC6A2
SCHEMBL23024527 0.68 OTUD7B (0.38) DRD2OPRD1BACE1OTUD7BPDK2
SCHEMBL24388827 0.68 DRD2 (0.41) DRD2OPRD1OPRK1BACE1OTUD7B
SCHEMBL30529476 0.68 OTUD7B (0.38) DRD2OPRD1BACE1OTUD7BPDK2
Hydrochloric Acid SCHEMBL23024386 0.67 OTUD7B (0.38) DRD2OPRD1BACE1OTUD7BPDK2
SCHEMBL21397337 0.66 HTR2A (0.37) SLC6A2SLC6A4
SCHEMBL21397254 0.65 DRD2 (0.32) DRD2
SCHEMBL13131168 0.64 ACHE (0.59) DRD2PDK2
SCHEMBL11931918 0.64 DRD2 (0.36) DRD2OPRD1BACE1OTUD7BPDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019183367-A1 SHP2 PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF RELAY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed