SCHEMBL21397675

SCHEMBL21397675

CCCC1(CCC)Cc2ccccc2C1NC

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.40
HRH1 P35367 3/20 0.40
PDPK1 O15530 1/20 0.38
SLC6A2 P23975 9/20 0.35
CYP2D6 P10635 8/20 0.35
SLC6A4 P31645 8/20 0.35
SLC6A3 Q01959 5/20 0.34
ADRA2A P08913 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
ADRA1B P35368 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21397337 0.77 HTR2A (0.37) HTR2AHRH1SLC6A2CYP2D6SLC6A4
SCHEMBL12086608 0.74 SLC10A2 (0.37) HTR2ASLC6A2CYP2D6SLC6A4ADRA2A
SCHEMBL21397653 0.74 HTR2A (0.35) HTR2AHRH1SLC6A2CYP2D6SLC6A4
SCHEMBL24388766 0.74 PDPK1 (0.47) HTR2AHRH1PDPK1SLC6A2CYP2D6
SCHEMBL2581679 0.74 PDPK1 (0.47) HTR2AHRH1PDPK1SLC6A2CYP2D6
SCHEMBL22515436 0.73 ALOX12 (0.38) ADRA2AADRA2BADRA2CADRA1B
SCHEMBL25522982 0.73 PDPK1 (0.42) HTR2AHRH1PDPK1SLC6A2CYP2D6
SCHEMBL22515488 0.72 MEN1 (0.38) CYP2D6ADRA2AADRA2BADRA2CADRA1B
SCHEMBL16448778 0.71 SLC6A2 (0.43) HTR2AHRH1PDPK1SLC6A2CYP2D6
SCHEMBL17559137 0.70 PDPK1 (0.40) HTR2AHRH1PDPK1SLC6A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019183367-A1 SHP2 PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF RELAY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed