SCHEMBL2139776

SCHEMBL2139776

[CH2]CCCCCCCCCC([CH2])CCCCCCCC

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.41
DNM1 Q05193 2/20 0.40
TSHR P16473 1/20 0.40
THRB P10828 1/20 0.40
OPRM1 P35372 1/20 0.39
GPR84 Q9NQS5 3/20 0.37
FDPS P14324 3/20 0.37
SPHK1 Q9NYA1 1/20 0.37
FFAR1 O14842 1/20 0.37
MAPT P10636 1/20 0.35
LCK P06239 1/20 0.35
PPARD Q03181 1/20 0.35
ZDHHC20 Q5W0Z9 1/20 0.35
ZDHHC2 Q9UIJ5 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2139902 1.00 LMNA (0.41) LMNADNM1TSHRTHRBOPRM1
SCHEMBL2140719 1.00 LMNA (0.41) LMNADNM1TSHRTHRBOPRM1
SCHEMBL2137295 1.00 LMNA (0.41) LMNADNM1TSHRTHRBOPRM1
SCHEMBL9656413 1.00 LMNA (0.41) LMNADNM1TSHRTHRBOPRM1
SCHEMBL1699698 1.00 LMNA (0.41) LMNADNM1TSHRTHRBOPRM1
SCHEMBL11285372 1.00 LMNA (0.41) LMNADNM1TSHRTHRBOPRM1
SCHEMBL3395197 1.00 LMNA (0.41) LMNADNM1TSHRTHRBOPRM1
SCHEMBL290240 1.00 LMNA (0.41) LMNADNM1TSHRTHRBOPRM1
SCHEMBL148380 0.95 DNM1 (0.40) LMNADNM1TSHRTHRBOPRM1
SCHEMBL19922801 0.95 DNM1 (0.40) LMNADNM1TSHRTHRBOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3394035-A1 USE OF SUBSTITUTED DIHYDROISOQUINOLINIUM SALTS FOR TREATING KERATIN MATERIALS, COMPOSITIONS AND IMPLEMENTATION PROCESSES L'Oréal (FR) 2018-10-31 EP disclosed
EP-3394034-A1 USE OF DIHYDROISOQUINOLINIUM SALTS FOR TREATING KERATIN MATERIALS, COMPOSITIONS AND IMPLEMENTATION PROCESSES L'Oréal (FR) 2018-10-31 EP disclosed
EP-1937734-B1 BIOCIDAL POLYMERS KE KELIT KUNSTSTOFFWERK GES M B H (AT) 2018-04-04 EP disclosed
WO-2017109185-A1 USE OF SUBSTITUTED DIHYDROISOQUINOLINIUM SALTS FOR TREATING KERATIN MATERIALS, COMPOSITIONS AND IMPLEMENTATION PROCESSES L'OREAL (FR) 2017-06-29 WO disclosed
WO-2017109183-A1 USE OF DIHYDROISOQUINOLINIUM SALTS FOR TREATING KERATIN MATERIALS, COMPOSITIONS AND IMPLEMENTATION PROCESSES L'OREAL (FR) 2017-06-29 WO disclosed
WO-2014118231-A2 DYE COMPOSITION USING AT LEAST ONE COUPLER OF META-AMINOPHENOL TYPE IN A MEDIUM COMPRISING A FATTY SUBSTANCE, PROCESSES AND DEVICE L'OREAL (FR) 2014-08-07 WO disclosed
EP-2707384-A1 CELL-REACTIVE, LONG-ACTING, OR TARGETED COMPSTATIN ANALOGS AND USES THEREOF Apellis Pharmaceuticals, Inc. (US) 2014-03-19 EP disclosed
EP-2542210-A2 COSMETIC ANTIDANDRUFF COMPOSITION BASED ON ELLAGIC ACID OR A DERIVATIVE THEREOF AND A SECOND, DIFFERENT ACTIVE COMPOUND IN A SPECIFIC WEIGHT RATIO L'Oréal (FR) 2013-01-09 EP disclosed
WO-2012155107-A1 CELL-REACTIVE, LONG-ACTING, OR TARGETED COMPSTATIN ANALOGS AND USES THEREOF APELLIS PHARMACEUTICALS, INC. (US) 2012-11-15 WO disclosed
US-8148484-B2 Poly(bicyclo[2.2.1]hept-5-ene-2-carboxylic acid 2-(tert-butylamino)ethyl ester); Poly(bicyclo[2.2.1]hept-5-ene-2-carboxylic acid 2-(dimethylamino)ethyl ester); used for disinfecting, sterilizing, and preventing biofouling in closed or open industrial-water systems and cooling-water systems KE KELIT KUNSTSTOFFWERK GESMBH (AT) 2012-04-03 US disclosed
WO-2011107468-A2 COSMETIC ANTIDANDRUFF COMPOSITION BASED ON ELLAGIC ACID OR A DERIVATIVE THEREOF AND A SECOND, DIFFERENT ACTIVE COMPOUND IN A SPECIFIC WEIGHT RATIO L'OREAL (FR) 2011-09-09 WO disclosed
US-20080251460-A1 Biocidal Polymers KE KELIT KUNSTSTOFFWERK GESMBH (AT) 2008-10-16 US disclosed
EP-1937734-A2 BIOCIDAL POLYMERS KE-KELIT Kunststoffwerk Gesellschaft m.b.H. (AT) 2008-07-02 EP disclosed
WO-2007045634-A2 BIOCIDAL POLYMERS KE KELIT KUNSTSTOFFWERK GESMBH (AT) 2007-04-26 WO disclosed
EP-0842196-A1 CELL ADHESION INHIBITORS BIOGEN, INC. (US) 1998-05-20 EP disclosed
WO-1995035088-A1 COSMETIC AND/OR PHARMACEUTICAL O/W EMULSIONS HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 1995-12-28 WO disclosed
US-5474778-A Contains at least one sterol ester in molecule; emulsifying and hydrating qualities AJINOMOTO CO., INC. (JP) 1995-12-12 US disclosed