SCHEMBL21409620

SCHEMBL21409620

O=C(c1ccc(Cl)cc1)c1cnn(-c2ccccc2)c1-c1ccc(Cl)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 2/20 0.55
LMNA P02545 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
ALDH1A1 P00352 1/20 0.51
RAB9A P51151 4/20 0.48
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
NPC1 O15118 3/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
NR4A1 P22736 1/20 0.48
PTGDR2 Q9Y5Y4 1/20 0.46
MAPT P10636 1/20 0.45
NFKB1 P19838 1/20 0.45
NFKB2 Q00653 1/20 0.45
RELA Q04206 1/20 0.45
PTGS2 P35354 2/20 0.44
CNR1 P21554 1/20 0.44
CNR2 P34972 1/20 0.44
KDM4E B2RXH2 1/20 0.44
GAA P10253 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7915015 0.87 MAPK14 (0.66) MAPK14NPSR1ALDH1A1MEN1KMT2A
SCHEMBL21409682 0.84 MAPK14 (0.56) MAPK14LMNANPSR1ALDH1A1RAB9A
SCHEMBL21409792 0.80 CNR1 (0.44) MAPK14LMNARAB9ANPC1NR4A1
SCHEMBL21409783 0.78 CNR1 (0.43) MAPK14LMNAALDH1A1MEN1KMT2A
SCHEMBL4497271 0.76 ALDH1A1 (0.65) MAPK14ALDH1A1RAB9AMEN1KMT2A
SCHEMBL11259925 0.76 KDM4E (0.54) LMNANPSR1ALDH1A1RAB9AMEN1
SCHEMBL8765024 0.75 RAB9A (0.69) LMNANPSR1ALDH1A1RAB9AMEN1
SCHEMBL11399825 0.75 LMNA (0.53) LMNANPSR1ALDH1A1RAB9AMEN1
SCHEMBL21409678 0.74 MAPK14 (0.45) MAPK14LMNANPSR1ALDH1A1MAPT
SCHEMBL21409788 0.74 CNR1 (0.53) MAPK14CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019188456-A1 NOVEL ANTI-TUMOR AGENT 学校法人 川崎学園 2019-10-03 WO disclosed