SCHEMBL21417606

SCHEMBL21417606

CN[C@H](Cc1ccc(N=O)cc1)C(C)=O

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FPR2 P25090 1/20 0.46
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37
NOS2 P35228 1/20 0.37
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
PPARG P37231 3/20 0.36
ALDH1A1 P00352 2/20 0.36
HSD17B10 Q99714 1/20 0.36
MME P08473 2/20 0.34
LMNA P02545 1/20 0.34
ACE P12821 1/20 0.33
CPA1 P15085 1/20 0.33
ACE2 Q9BYF1 1/20 0.33
EPHX1 P07099 1/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
FOLH1 Q04609 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL805214 0.87 FPR2 (0.56) FPR2PPARGMMELMNAACE
SCHEMBL25101017 0.84 FPR2 (0.44) FPR2NOS3NOS1NOS2ESR1
SCHEMBL8231892 0.81 ESR1 (0.56) ESR1ESR2MMEACECPA1
SCHEMBL16327905 0.81 ESR1 (0.40) NOS3NOS1ESR1ESR2PPARG
SCHEMBL12668874 0.81 ACACB (0.46) ESR1ESR2PPARGALDH1A1
SCHEMBL9886030 0.81 ACACB (0.46) ESR1ESR2PPARGALDH1A1
SCHEMBL14942927 0.81 ESR1 (0.56) ESR1ESR2MMEACECPA1
SCHEMBL7637685 0.81 ESR1 (0.56) ESR1ESR2MMEACECPA1
SCHEMBL24329157 0.79 ACACB (0.48) FPR2MMEEPHX1CTSSCTSK
SCHEMBL12668867 0.79 ACACB (0.48) FPR2MMEEPHX1CTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2316846-B1 Spatially-defined macrocyclic compounds useful for drug discovery OCERA THERAPEUTICS INC (US) 2019-10-02 EP disclosed