SCHEMBL2142185

SCHEMBL2142185

O=C(O)N1CCC2(CC1)CN(C(=O)C(F)(F)F)CCO2

nearest known ligand 0.45

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 14/20 0.45
MGLL Q99685 6/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18422101 0.85 CHRM2 (0.42) EPHX2MGLL
SCHEMBL10241579 0.82 EPHX2 (0.40) EPHX2MGLL
Trifluoroacetic Acid SCHEMBL1246075 0.81 EPHX2 (0.38) EPHX2MGLL
SCHEMBL2142168 0.81 USP2 (0.49) EPHX2MGLL
SCHEMBL19097004 0.76 EPHX2 (0.44) EPHX2
SCHEMBL30545528 0.75 CHRM2 (0.39) EPHX2MGLL
SCHEMBL18341792 0.74 VNN1 (0.37) EPHX2MGLL
SCHEMBL31548277 0.74 CNR2 (0.37) EPHX2MGLL
SCHEMBL17318867 0.72 CHRM2 (0.65) EPHX2MGLL
SCHEMBL30900658 0.72 VNN1 (0.38) EPHX2MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8629271-B2 Compounds ASTRAZENECA AB (GB) 2014-01-14 US disclosed
US-20120322788-A1 Compouds PULMAGEN THERAPEUTICS (SYNERGY) LIMITED (GB) 2012-12-20 US disclosed
EP-2242759-B1 COMPOUNDS ASTRAZENECA AB (SE) 2012-09-12 EP disclosed
US-8148373-B2 Compounds ASTRAZENECA AB (SE) 2012-04-03 US disclosed
EP-2242759-A1 COMPOUNDS AstraZeneca AB (SE) 2010-10-27 EP disclosed
US-20090298807-A1 Compounds ASTRAZENECA AB (SE) 2009-12-03 US disclosed
WO-2009098448-A1 COMPOUNDS ASTRAZENECA AB (SE) 2009-08-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120322788-A1 Compouds PKD1, SBDS, ABCB11 EPHX2 1056/4885MGLL 4101/4885
US-20090298807-A1 Compounds PKD1, SLC10A1, ABCB11 EPHX2 1481/4885MGLL 3335/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.