SCHEMBL2145157

SCHEMBL2145157

CCc1cc(NC(=O)Nc2ccc(Cn3cnc(O)c3C(N)=O)cc2)ccc1C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.39
RAB9A P51151 3/20 0.36
NPC1 O15118 2/20 0.36
TP53 P04637 1/20 0.36
POLB P06746 1/20 0.36
FGFR1 P11362 2/20 0.36
FGFR4 P22455 2/20 0.36
ITGB1 P05556 2/20 0.36
ITGA4 P13612 2/20 0.36
PKM P14618 1/20 0.35
MITF O75030 1/20 0.35
PAX8 Q06710 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MEN1 O00255 1/20 0.35
USP2 O75604 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2145497 0.86 RAB9A (0.49) RAB9ANPC1TP53POLBFGFR1
SCHEMBL2145359 0.84 MEN1 (0.44) NR1I2TP53POLBITGB1ITGA4
SCHEMBL2145723 0.84 NPC1 (0.52) NR1I2RAB9ANPC1POLBMITF
SCHEMBL2145641 0.83 RAB9A (0.46) NR1I2RAB9ANPC1TP53POLB
SCHEMBL2145819 0.83 KDM4E (0.41) NR1I2RAB9ANPC1TP53POLB
SCHEMBL2145339 0.82 NR1I2 (0.46) NR1I2RAB9ANPC1POLBITGB1
SCHEMBL2145716 0.81 GHSR (0.42) RAB9ANPC1FGFR1FGFR4SMN1; SMN2
SCHEMBL13651666 0.81 KMT2A (0.46) FGFR1FGFR4PKMALDH1A1TSHR
SCHEMBL2145865 0.81 MEN1 (0.43) RAB9ANPC1POLBFGFR1FGFR4
SCHEMBL2145460 0.81 SAE1 (0.55) RAB9ANPC1FGFR1PKMSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2040702-B1 USE OF AMPK-ACTIVATING IMIDAZOLE DERIVATIVES, PREPARATION PROCESS THEREFOR AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM MERCK PATENT GMBH (DE) 2011-07-27 EP claimed