SCHEMBL21452003

SCHEMBL21452003

CN(C(=O)OC(C)(C)C)C1(c2ccc(C(F)(F)F)c(C#N)c2)CCCCC1=O

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AR P10275 9/20 0.34
CACNA1G O43497 1/20 0.34
CACNA1B Q00975 1/20 0.34
CACNA1C Q13936 1/20 0.34
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
TACR1 P25103 1/20 0.33
CYP2C19 P33261 1/20 0.33
KCNH2 Q12809 1/20 0.33
SLC22A12 Q96S37 1/20 0.32
PDE2A O00408 3/20 0.31
BCL2A1 Q16548 1/20 0.31
TSHR P16473 1/20 0.30
KCNN4 O15554 1/20 0.30
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21452251 0.79 TRPA1 (0.36) ARCYP2D6CYP2C9TACR1CYP2C19
SCHEMBL21452535 0.77 GAA (0.40) CACNA1GCACNA1BCACNA1CCYP2C9CYP2C19
SCHEMBL21452009 0.75 CYP11B2 (0.38) CYP2C9CYP2C19TSHR
SCHEMBL21452002 0.73 SLC22A12 (0.38) ARCYP2D6CYP2C9TACR1CYP2C19
SCHEMBL21452004 0.73 SLC22A12 (0.38) ARCYP2D6CYP2C9TACR1CYP2C19
SCHEMBL21452538 0.70 SLC22A12 (0.34) ARCYP2D6CYP2C9TACR1CYP2C19
SCHEMBL21452005 0.69 CYP2D6 (0.35) ARCYP2D6CYP2C9TACR1CYP2C19
SCHEMBL26451021 0.68 TSHR (0.61) CACNA1CCYP2C9CYP2C19TSHR
SCHEMBL21452447 0.64 PDE2A (0.43) PDE2AKCNN4
SCHEMBL21436244 0.63 AR (0.34) ARCYP2D6CYP2C9TACR1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3778579-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Jianhe Pharmaceutical & Technology Co. Ltd. (CN) 2021-02-17 EP disclosed
WO-2019192602-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海键合医药科技有限公司 2019-10-10 WO disclosed