SCHEMBL21452002

SCHEMBL21452002

N#Cc1cc(C2(Cl)CCCCC2=O)ccc1C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 1/20 0.38
PDE2A O00408 1/20 0.35
AR P10275 14/20 0.34
TRPA1 O75762 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
TACR1 P25103 1/20 0.34
CYP2C19 P33261 1/20 0.34
KCNH2 Q12809 1/20 0.34
PGR P06401 1/20 0.32
RXRA P19793 1/20 0.32
RXRB P28702 1/20 0.32
RXRG P48443 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21452004 0.85 SLC22A12 (0.38) SLC22A12PDE2AARTRPA1CYP2D6
SCHEMBL23490891 0.82 CYP11B2 (0.33)
SCHEMBL21452511 0.81 HDAC1 (0.45) PDE2AAR
SCHEMBL21452538 0.79 SLC22A12 (0.34) SLC22A12PDE2AARTRPA1CYP2D6
SCHEMBL21452416 0.75 SLC6A3 (0.44) PDE2A
SCHEMBL21452022 0.75 CYP19A1 (0.40) CYP2D6PGR
SCHEMBL21452251 0.74 TRPA1 (0.36) SLC22A12PDE2AARTRPA1CYP2D6
SCHEMBL21452525 0.73 PGR (0.40) PGR
SCHEMBL21452498 0.69 HDAC4 (0.35) AR
SCHEMBL21451899 0.68 TACR1 (0.41) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210171487-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF SHANGHAI JIANHE PHARMACEUTICAL & TECHNOLOGY CO. LTD. (CN) 2021-06-10 US disclosed
EP-3778579-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Jianhe Pharmaceutical & Technology Co. Ltd. (CN) 2021-02-17 EP disclosed
WO-2019192602-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海键合医药科技有限公司 2019-10-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210171487-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF CYP4F11, PAH, COMT SLC22A12 692/4885PDE2A 4338/4885AR 1775/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.