SCHEMBL21452010

SCHEMBL21452010

N#Cc1ccc(C2CCCCC2=O)c(F)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 9/20 0.50
CYP11B1 P15538 4/20 0.50
CYP19A1 P11511 2/20 0.50
CYP17A1 P05093 1/20 0.44
HRH1 P35367 1/20 0.44
KCNH2 Q12809 1/20 0.44
ELANE P08246 1/20 0.38
HSD11B1 P28845 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.34
CHRNA1 P02708 1/20 0.34
CHRNG P07510 1/20 0.34
CHRNB1 P11230 1/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA4 P43681 1/20 0.34
CHRND Q07001 1/20 0.34
AURKA O14965 1/20 0.33
DAPK3 O43293 1/20 0.33
PRKD3 O94806 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19993831 0.78 OPRL1 (0.42) TLR4KMT2A
SCHEMBL21452585 0.77 DRD2 (0.49) KMT2AMCOLN3
SCHEMBL27219407 0.75 DRD2 (0.48) KMT2AMCOLN3
SCHEMBL5071326 0.75 CYP19A1 (0.43) CYP11B2CYP11B1CYP19A1KCNH2TLR4
SCHEMBL16839687 0.75 CYP11B2 (0.50) CYP11B2CYP11B1CYP19A1CYP17A1HRH1
SCHEMBL360459 0.75 TP53 (0.42) CYP11B2CYP17A1TLR4KMT2A
SCHEMBL28770987 0.75 IDO1 (0.61)
SCHEMBL29671045 0.75 IDO1 (0.61)
SCHEMBL19993936 0.74 MAPK1 (0.46)
SCHEMBL10356725 0.73 KDM4E (0.45) CYP19A1TLR4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210171487-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF SHANGHAI JIANHE PHARMACEUTICAL & TECHNOLOGY CO. LTD. (CN) 2021-06-10 US disclosed
EP-3778579-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Jianhe Pharmaceutical & Technology Co. Ltd. (CN) 2021-02-17 EP disclosed
WO-2019192602-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海键合医药科技有限公司 2019-10-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210171487-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF CYP4F11, PAH, COMT CYP11B2 18/4885CYP11B1 15/4885CYP19A1 386/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.