SCHEMBL21452012

SCHEMBL21452012

N#Cc1ccc(C2(N)CCCCC2=O)c(F)c1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.42
CYP11B2 P19099 3/20 0.38
PGR P06401 5/20 0.35
DRD2 P14416 2/20 0.34
DRD3 P35462 2/20 0.34
PNMT P11086 1/20 0.34
CYP11B1 P15538 2/20 0.34
HSD11B1 P28845 1/20 0.34
CYP19A1 P11511 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
BACE1 P56817 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21452011 0.81 CYP11B2 (0.38) KDM1ACYP11B2PGRCYP11B1HSD11B1
SCHEMBL21451916 0.79 KDM1A (0.38) KDM1A
SCHEMBL21452509 0.77 P2RX7 (0.39) KDM1ACYP11B2CYP11B1CYP19A1BACE1
SCHEMBL21452018 0.77 CYP19A1 (0.40) KDM1ACYP11B2PGRCYP19A1MAOA
SCHEMBL21452013 0.75 CYP11B2 (0.35) KDM1ACYP11B2PGRCYP11B1HSD11B1
SCHEMBL27173461 0.75 HDAC4 (0.47) KDM1AHSD11B1
SCHEMBL21452474 0.75 ABCC9 (0.40) KDM1APGRHSD11B1MAOAMAOB
SCHEMBL21452504 0.71 KDM1A (0.40) KDM1A
SCHEMBL24815346 0.70 HDAC4 (0.51) KDM1A
SCHEMBL16014962 0.70 KDM1A (0.45) KDM1ADRD2DRD3PNMTBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210171487-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF SHANGHAI JIANHE PHARMACEUTICAL & TECHNOLOGY CO. LTD. (CN) 2021-06-10 US disclosed
EP-3778579-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Jianhe Pharmaceutical & Technology Co. Ltd. (CN) 2021-02-17 EP disclosed
WO-2019192602-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海键合医药科技有限公司 2019-10-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210171487-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF CYP4F11, PAH, COMT KDM1A 3700/4885CYP11B2 18/4885PGR 3651/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.