SCHEMBL2145821

SCHEMBL2145821

CC(C)(C)N1CCC(C(=O)c2cccc(F)c2)C1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 5/20 0.53
KMT2A Q03164 4/20 0.53
MEN1 O00255 2/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
MGLL Q99685 2/20 0.50
ALDH1A1 P00352 3/20 0.47
HTR1F P30939 1/20 0.45
EPHX2 P34913 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4975598 0.92 MEN1 (0.53) HSD11B1KMT2AMEN1CYP2C9CYP2C19
SCHEMBL23022742 0.92 HSD11B1 (0.59) HSD11B1KMT2AMEN1CYP2C9CYP2C19
SCHEMBL5316077 0.83 KMT2A (0.53) HSD11B1KMT2AMEN1MGLLALDH1A1
SCHEMBL2146383 0.79 HSD11B1 (0.54) HSD11B1KMT2AMEN1CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL10640478 0.78 KMT2A (0.65) HSD11B1KMT2AMEN1CYP2C9CYP2C19
SCHEMBL3965621 0.77 KDM2B (0.66) KMT2AMEN1ALDH1A1
SCHEMBL3895577 0.75 HSD11B1 (0.69) HSD11B1KMT2AMEN1CYP2C9CYP2C19
SCHEMBL5475032 0.75 ALDH1A1 (0.59) KMT2AMEN1ALDH1A1
SCHEMBL969184 0.75 ALDH1A1 (0.59) KMT2AMEN1ALDH1A1
SCHEMBL969182 0.75 ALDH1A1 (0.59) KMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011088045-A1 AURORA KINASE COMPOUNDS AND METHODS OF THEIR USE AMBIT BIOSCIENCES CORPORATION (US) 2011-07-21 WO disclosed