SCHEMBL4975598

SCHEMBL4975598

CC(C)(C)N1CCC[C@@H](C(=O)c2cccc(F)c2)C1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
ALDH1A1 P00352 1/20 0.53
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
HSD11B1 P28845 1/20 0.48
KDM2B Q8NHM5 11/20 0.47
MGLL Q99685 1/20 0.46
KDM4E B2RXH2 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2145821 0.92 HSD11B1 (0.53) MEN1KMT2AALDH1A1CYP2C9CYP2C19
SCHEMBL3965621 0.85 KDM2B (0.66) MEN1KMT2AALDH1A1KDM2B
SCHEMBL23022742 0.84 HSD11B1 (0.59) MEN1KMT2AALDH1A1CYP2C9CYP2C19
SCHEMBL4079510 0.81 KDM2B (0.44) MEN1KMT2AALDH1A1KDM2BMGLL
SCHEMBL969184 0.80 ALDH1A1 (0.59) MEN1KMT2AALDH1A1
SCHEMBL5475032 0.80 ALDH1A1 (0.59) MEN1KMT2AALDH1A1
SCHEMBL27778359 0.80 KMT2A (0.52) MEN1KMT2AALDH1A1CYP2C9CYP2C19
SCHEMBL969182 0.80 ALDH1A1 (0.59) MEN1KMT2AALDH1A1
SCHEMBL4082779 0.80 ALDH1A1 (0.61) MEN1KMT2AALDH1A1CYP2C9CYP2C19
SCHEMBL23579339 0.78 HSD11B1 (0.58) MEN1KMT2AALDH1A1CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1966139-A1 ASPARTIC PROTEASE INHIBITORS Vitae Pharmaceuticals, Inc. (US) 2008-09-10 EP disclosed
WO-2007070201-A1 ASPARTIC PROTEASE INHIBITORS VITAE PHARMACEUTICALS, INC. (US) 2007-06-21 WO disclosed