SCHEMBL2146188

SCHEMBL2146188

O=C(CCl)Nc1ccc(Sc2nc(Nc3cc(C4CC4)[nH]n3)n3cccc3n2)cc1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 17/20 0.51
SRC P12931 4/20 0.51
GSK3B P49841 2/20 0.51
AURKA O14965 13/20 0.46
AURKC Q9UQB9 5/20 0.43
ABL1 P00519 1/20 0.41
YES1 P07947 1/20 0.41
HCK P08631 1/20 0.41
CCNE2 O96020 1/20 0.39
IGF1R P08069 1/20 0.39
CCNE1 P24864 1/20 0.39
CDK2 P24941 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2148571 0.97 AURKB (0.48) AURKBSRCGSK3BAURKAAURKC
SCHEMBL2146309 0.87 AURKB (0.55) AURKBSRCGSK3BAURKAAURKC
SCHEMBL2148602 0.85 AURKB (0.58) AURKBSRCGSK3BAURKAAURKC
SCHEMBL2149372 0.85 AURKB (0.48) AURKBSRCGSK3BAURKA
SCHEMBL2148687 0.85 AURKB (0.41) AURKBSRCGSK3BAURKAAURKC
SCHEMBL2148465 0.85 AURKB (0.43) AURKBSRCGSK3BAURKAAURKC
SCHEMBL2183054 0.84 AURKB (0.58) AURKBSRCGSK3BAURKAAURKC
SCHEMBL2146695 0.84 AURKB (0.58) AURKBSRCGSK3BAURKAAURKC
SCHEMBL2153217 0.84 SRC (0.44) AURKBSRCGSK3BAURKACCNE2
SCHEMBL2148475 0.82 NPC1 (0.43) AURKBSRCGSK3BAURKAAURKC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011088045-A1 AURORA KINASE COMPOUNDS AND METHODS OF THEIR USE AMBIT BIOSCIENCES CORPORATION (US) 2011-07-21 WO disclosed