SCHEMBL2148571

SCHEMBL2148571

O=C(CCl)Nc1ccc(Sc2nc(Nc3cc(C4CCC4)[nH]n3)n3cccc3n2)cc1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 19/20 0.48
SRC P12931 1/20 0.48
GSK3B P49841 1/20 0.48
AURKA O14965 17/20 0.43
AURKC Q9UQB9 5/20 0.43
LCK P06239 1/20 0.41
ITK Q08881 1/20 0.41
NTRK1 P04629 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2146188 0.97 AURKB (0.51) AURKBSRCGSK3BAURKAAURKC
SCHEMBL2146309 0.85 AURKB (0.55) AURKBSRCGSK3BAURKAAURKC
SCHEMBL2203289 0.84 AURKA (0.47) AURKBSRCGSK3BAURKALCK
SCHEMBL2161764 0.84 AURKB (0.57) AURKBSRCGSK3BAURKAAURKC
SCHEMBL2148602 0.84 AURKB (0.58) AURKBSRCGSK3BAURKAAURKC
SCHEMBL2148687 0.83 AURKB (0.41) AURKBSRCGSK3BAURKAAURKC
SCHEMBL2148465 0.83 AURKB (0.43) AURKBSRCGSK3BAURKAAURKC
SCHEMBL2149372 0.82 AURKB (0.48) AURKBSRCGSK3BAURKA
SCHEMBL2183054 0.81 AURKB (0.58) AURKBSRCGSK3BAURKAAURKC
SCHEMBL2148475 0.81 NPC1 (0.43) AURKBSRCGSK3BAURKAAURKC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011088045-A1 AURORA KINASE COMPOUNDS AND METHODS OF THEIR USE AMBIT BIOSCIENCES CORPORATION (US) 2011-07-21 WO disclosed