SCHEMBL2146295

SCHEMBL2146295

O=C(c1cccc(F)c1)C1CCNC1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.50
CES2 O00748 1/20 0.49
CES1 P23141 1/20 0.49
KMT2A Q03164 3/20 0.47
MEN1 O00255 2/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
MGLL Q99685 1/20 0.47
PARP1 P09874 1/20 0.46
GRM5 P41594 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
CDK5 Q00535 2/20 0.43
CDK5R1 Q15078 2/20 0.43
CYP2D6 P10635 1/20 0.43
PLA2G7 Q13093 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12023170 0.93 CDK5 (0.47) HSD11B1CES2CES1KMT2AMEN1
SCHEMBL3957507 0.93 CDK5 (0.47) HSD11B1CES2CES1KMT2AMEN1
Hydrochloric Acid SCHEMBL5476502 0.91 CDK5 (0.47) HSD11B1CES2CES1KMT2AMEN1
Hydrochloric Acid SCHEMBL5476506 0.91 CDK5 (0.47) HSD11B1CES2CES1KMT2AMEN1
SCHEMBL11620780 0.90 HSD11B1 (0.56) HSD11B1CES2CES1KMT2AMEN1
Hydrochloric Acid SCHEMBL15566694 0.89 KMT2A (0.55) HSD11B1CES2CES1KMT2AMEN1
SCHEMBL9923375 0.89 CES2 (0.53) HSD11B1CES2CES1KMT2AMEN1
SCHEMBL2146518 0.82 MEN1 (0.54) HSD11B1KMT2AMEN1MGLLCYP2D6
SCHEMBL407286 0.82 KMT2A (0.53) HSD11B1KMT2AMEN1MGLLCYP2D6
SCHEMBL30577937 0.81 PARP1 (0.43) KMT2AMEN1PARP1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011088045-A1 AURORA KINASE COMPOUNDS AND METHODS OF THEIR USE AMBIT BIOSCIENCES CORPORATION (US) 2011-07-21 WO disclosed