SCHEMBL9923375

SCHEMBL9923375

O=C(c1cccc(F)c1)C1CNC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.53
CES1 P23141 2/20 0.53
CYP2C9 P11712 2/20 0.50
CYP2C19 P33261 2/20 0.50
PARP1 P09874 1/20 0.50
HSD11B1 P28845 1/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
HDAC1 Q13547 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
MGLL Q99685 1/20 0.47
PLA2G7 Q13093 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.45
GRM5 P41594 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
ALDH1A1 P00352 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
CYP1A2 P05177 1/20 0.42
GAA P10253 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2146295 0.89 HSD11B1 (0.50) CES2CES1CYP2C9CYP2C19PARP1
SCHEMBL11620780 0.85 HSD11B1 (0.56) CES2CES1CYP2C9CYP2C19PARP1
SCHEMBL3957507 0.85 CDK5 (0.47) CES2CES1CYP2C9CYP2C19PARP1
SCHEMBL12023170 0.85 CDK5 (0.47) CES2CES1CYP2C9CYP2C19PARP1
Hydrochloric Acid SCHEMBL5476502 0.84 CDK5 (0.47) CES2CES1CYP2C9CYP2C19PARP1
Hydrochloric Acid SCHEMBL5476506 0.84 CDK5 (0.47) CES2CES1CYP2C9CYP2C19PARP1
Hydrochloric Acid SCHEMBL15566694 0.83 KMT2A (0.55) CES2CES1CYP2C9CYP2C19PARP1
SCHEMBL1528775 0.82 CES2 (0.46) CES2CES1HSD11B1MEN1KMT2A
SCHEMBL23579339 0.81 HSD11B1 (0.58) CES2CES1CYP2C9CYP2C19PARP1
SCHEMBL29973506 0.81 HSD11B1 (0.58) CES2CES1CYP2C9CYP2C19PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012076063-A1 PYRIDINE AMIDE DERIVATIVES AS EP4 RECEPTOR ANTAGONISTS ROTTAPHARM S.P.A. (IT) 2012-06-14 WO disclosed