SCHEMBL21469191

SCHEMBL21469191

CC(=O)N1CCc2cc(Br)c(S(=O)(=O)N(C)CI)cc21

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
XIAP P98170 2/20 0.49
BIRC2 Q13490 2/20 0.49
ACLY P53396 1/20 0.48
NOTUM Q6P988 5/20 0.42
LMNA P02545 3/20 0.42
TSHR P16473 1/20 0.42
ALDH1A1 P00352 2/20 0.41
MEN1 O00255 1/20 0.41
HPGD P15428 1/20 0.41
KMT2A Q03164 1/20 0.41
IDO1 P14902 1/20 0.40
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TRIM24 O15164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17545148 0.89 XIAP (0.53) XIAPBIRC2ACLYNOTUMLMNA
SCHEMBL17545284 0.83 MEN1 (0.62) XIAPBIRC2ACLYLMNAALDH1A1
SCHEMBL17545341 0.83 LMNA (0.49) XIAPBIRC2ACLYNOTUMLMNA
SCHEMBL17545102 0.82 NOTUM (0.49) XIAPBIRC2ACLYNOTUMLMNA
SCHEMBL17545361 0.81 TSHR (0.59) XIAPBIRC2ACLYNOTUMLMNA
SCHEMBL5332602 0.81 ACLY (0.53) XIAPBIRC2ACLYNOTUMLMNA
SCHEMBL14058949 0.81 ACLY (0.53) XIAPBIRC2ACLYNOTUMALDH1A1
SCHEMBL29707967 0.80 ACLY (0.53) XIAPBIRC2ACLYNOTUMALDH1A1
SCHEMBL1179278 0.80 ACLY (0.53) XIAPBIRC2ACLYNOTUMALDH1A1
SCHEMBL17545314 0.78 TSHR (0.46) XIAPBIRC2ACLYNOTUMLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3180312-B1 INDOLINE SULFONAMIDE INHIBITORS OF DAPE AND NDM-1 AND USE OF THE SAME UNIV LOYOLA CHICAGO (US) 2019-10-16 EP disclosed