SCHEMBL21473086

SCHEMBL21473086

C/C=C\c1ccc([N+](=O)[O-])cc1C

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.58
TSHR P16473 4/20 0.58
TDP1 Q9NUW8 3/20 0.58
CYP3A4 P08684 5/20 0.55
LMNA P02545 2/20 0.45
HTT P42858 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
ACHE P22303 2/20 0.44
HSD17B10 Q99714 1/20 0.44
TXNRD1 Q16881 1/20 0.43
TXNRD3 Q86VQ6 1/20 0.43
TXNRD2 Q9NNW7 1/20 0.43
MAPT P10636 3/20 0.43
KMT2A Q03164 2/20 0.43
MAPK1 P28482 1/20 0.43
ERN1 O75460 1/20 0.42
CRHBP P24387 2/20 0.42
CRHR2 Q13324 2/20 0.42
NFE2L2 Q16236 1/20 0.41
PDE2A O00408 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17199072 0.86 ALDH1A1 (0.58) ALDH1A1TSHRTDP1CYP3A4LMNA
SCHEMBL19623140 0.82 ALDH1A1 (0.58) ALDH1A1TSHRTDP1CYP3A4LMNA
SCHEMBL1858387 0.81 ALDH1A1 (0.62) ALDH1A1TSHRTDP1CYP3A4LMNA
SCHEMBL13696015 0.81 ALDH1A1 (0.59) ALDH1A1TSHRTDP1CYP3A4LMNA
SCHEMBL31415237 0.81 ALDH1A1 (0.44) ALDH1A1TSHRTDP1CYP3A4LMNA
SCHEMBL11343653 0.81 CYP3A4 (0.56) ALDH1A1TSHRTDP1CYP3A4LMNA
SCHEMBL10850493 0.80 ALDH1A1 (0.51) ALDH1A1TSHRTDP1CYP3A4LMNA
SCHEMBL10850498 0.80 ALDH1A1 (0.51) ALDH1A1TSHRTDP1CYP3A4LMNA
SCHEMBL28069165 0.80 NFE2L2 (0.61) ALDH1A1TSHRTDP1CYP3A4LMNA
SCHEMBL7134052 0.80 PTGES (0.59) ALDH1A1TSHRTDP1CYP3A4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3216787-B1 INTERMEDIATES FOR THE PREPARATION OF MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMA (US) 2020-02-19 EP disclosed
WO-2019200224-A1 SYNERGISTIC DRUG COMBINATIONS PREDICTED FROM GENOMIC FEATURES AND SINGLE-AGENT RESPONSE PROFILES THE BROAD INSTITUTE, INC. (US) 2019-10-17 WO disclosed