SCHEMBL21473592

SCHEMBL21473592

CCC(c1cccc(F)c1)N1Cc2ccccc2C1=O

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.55
KMT2A Q03164 5/20 0.55
MAPT P10636 5/20 0.48
TDP1 Q9NUW8 2/20 0.48
ALOX15 P16050 2/20 0.47
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
TSHR P16473 1/20 0.47
XIAP P98170 1/20 0.47
HKDC1 Q2TB90 1/20 0.47
HSD17B10 Q99714 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
TP53 P04637 1/20 0.46
THRB P10828 3/20 0.45
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22997449 0.86 MEN1 (0.59) MEN1KMT2AMAPTTDP1ALOX15
SCHEMBL6289218 0.78 TP53 (0.60) MEN1KMT2AMAPTTP53
SCHEMBL6287582 0.78 TP53 (0.60) MEN1KMT2AMAPTTP53
SCHEMBL4856275 0.78 TP53 (0.60) MEN1KMT2AMAPTTP53
SCHEMBL29419401 0.77 MEN1 (0.73) MEN1KMT2AMAPTTDP1ALOX15
SCHEMBL30046742 0.77 ALOX15 (0.59) MEN1KMT2AMAPTTDP1ALOX15
SCHEMBL21473668 0.76 THRB (0.61) MAPTTDP1ALOX15KDM4EALDH1A1
SCHEMBL23424735 0.75 ALOX15 (0.45) MEN1KMT2AMAPTTDP1ALOX15
SCHEMBL27679834 0.74 SLC6A2 (0.60) MAPTTP53THRB
SCHEMBL23424771 0.74 THRB (0.57) MAPTTDP1ALOX15KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019196938-A1 QUINAZOLINE COMPOUND SERVING AS EGFR TRIPLE MUTATION INHIBITOR AND APPLICATIONS THEREOF 华东理工大学 2019-10-17 WO disclosed