SCHEMBL21473717

SCHEMBL21473717

COC(=O)CCc1c(C)cc(C#N)cc1C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.45
PDE3A Q14432 1/20 0.45
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
TSHR P16473 5/20 0.39
HTT P42858 1/20 0.39
MAPK1 P28482 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HPGD P15428 4/20 0.38
HSD17B10 Q99714 4/20 0.38
ALDH1A1 P00352 3/20 0.38
GPR35 Q9HC97 2/20 0.38
TP53 P04637 2/20 0.38
MAPT P10636 1/20 0.38
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
EGFR P00533 1/20 0.37
SRC P12931 1/20 0.37
MEN1 O00255 1/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6829455 0.83 HSP90AB1 (0.41) TSHRHTTSMN1; SMN2HPGDHSD17B10
SCHEMBL1187327 0.83 ALDH1A1 (0.38) ALDH1A1GPR35MAPTMEN1KMT2A
SCHEMBL1969526 0.81 FFAR1 (0.50) TSHRHPGDHSD17B10ALDH1A1MEN1
SCHEMBL5990756 0.80 HSP90AB1 (0.47) PDE3BPDE3ATSHRHTTMAPK1
SCHEMBL1175089 0.78 CYP4F2 (0.41) TSHRHPGDHSD17B10ALDH1A1GPR35
SCHEMBL28407881 0.77 MAPT (0.43) TSHRHTTHPGDHSD17B10ALDH1A1
SCHEMBL6832152 0.77 GPR35 (0.38) TSHRHTTSMN1; SMN2HPGDHSD17B10
SCHEMBL2154006 0.76 TTR (0.39) TSHRALDH1A1GPR35MEN1KMT2A
SCHEMBL15061431 0.75 NOS3 (0.38) HPGDGPR35MAPTGAARAB9A
SCHEMBL3208670 0.75 ALDH1A1 (0.34) ALDH1A1GPR35CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019197274-A1 PROCESS FOR THE PREPARATION OF OPIOID MODULATORS QUIMICA SINTETICA, S. A. (ES) 2019-10-17 WO disclosed