SCHEMBL21484069

SCHEMBL21484069

N#Cc1ccccc1-n1cc(Br)cn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CREBBP Q92793 2/20 0.41
KDM4E B2RXH2 1/20 0.40
BRD4 O60885 1/20 0.39
PRKCI P41743 1/20 0.39
ERCC5 P28715 1/20 0.38
FEN1 P39748 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HIF1A Q16665 1/20 0.38
SLC2A1 P11166 1/20 0.37
SLC2A2 P11168 1/20 0.37
SLC2A3 P11169 1/20 0.37
HTR1A P08908 1/20 0.36
ADRA1D P25100 1/20 0.36
ADRA1A P35348 1/20 0.36
ADRA1B P35368 1/20 0.36
PTGES O14684 1/20 0.35
AXL P30530 1/20 0.35
GRM5 P41594 1/20 0.35
MAPT P10636 1/20 0.35
TSHR P16473 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23381882 0.80 CREBBP (0.41) CREBBPKDM4EBRD4ERCC5FEN1
SCHEMBL21877551 0.80 BRD4 (0.42) CREBBPKDM4EBRD4ERCC5FEN1
SCHEMBL27748840 0.80 TDO2 (0.41) CREBBPKDM4EBRD4ERCC5FEN1
SCHEMBL20738212 0.80 KDM4E (0.46) CREBBPKDM4EBRD4ERCC5FEN1
SCHEMBL24352877 0.78 CYP3A4 (0.43) CREBBPKDM4EBRD4ERCC5FEN1
SCHEMBL21706148 0.76 CREBBP (0.41) CREBBPKDM4EBRD4ERCC5FEN1
SCHEMBL31055062 0.76 ERCC5 (0.45) CREBBPKDM4EBRD4ERCC5FEN1
SCHEMBL31055053 0.76 CREBBP (0.41) CREBBPKDM4EBRD4ERCC5FEN1
SCHEMBL30607652 0.76 CREBBP (0.41) CREBBPKDM4EBRD4ERCC5FEN1
SCHEMBL24908426 0.75 CREBBP (0.38) CREBBPKDM4EBRD4ERCC5FEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019197549-A1 PYRAZOLO-TRIAZINE AND/OR PYRAZOLO-PYRIMIDINE DERIVATIVES AS SELECTIVE INHIBITOR OF CYCLIN DEPENDENT KINASE QURIENT CO., LTD. (KR) 2019-10-17 WO disclosed