SCHEMBL21494778

SCHEMBL21494778

CCNc1cccc2nn(C)cc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
USP2 O75604 1/20 0.40
CASP1 P29466 1/20 0.40
BRCA1 P38398 1/20 0.40
CASP7 P55210 1/20 0.40
SYK P43405 7/20 0.39
IDO1 P14902 2/20 0.39
ADORA3 P0DMS8 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA2B P29275 1/20 0.38
ADORA1 P30542 1/20 0.38
USP7 Q93009 1/20 0.37
POLB P06746 2/20 0.36
MAT2A P31153 1/20 0.36
NPC1 O15118 1/20 0.35
MAPT P10636 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
BRD4 O60885 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10933576 0.83 CA12 (0.49) SYKIDO1ADORA3ADORA2AADORA1
SCHEMBL19440644 0.81 SYK (0.37) MEN1KMT2AUSP2SYKADORA3
SCHEMBL28866124 0.75 PABPC1 (0.38) SYKPOLBMAPTBRD4CREBBP
SCHEMBL17680609 0.74 USP7 (0.41) USP7POLBMAPTBRD4CREBBP
SCHEMBL16775248 0.71 CREBBP (0.38) ADORA3ADORA1USP7POLBNPC1
SCHEMBL7946910 0.71 CYP2A6 (0.42) MEN1KMT2AADORA3ADORA2AADORA1
SCHEMBL11061959 0.70 ADRA2A (0.47) SYK
SCHEMBL19539233 0.69 BRD4 (0.40) USP7MAPTBRD4CREBBP
SCHEMBL8538647 0.69 KDM4E (0.41) ADORA2AADORA1USP7POLBNPC1
SCHEMBL17547027 0.69 CREBBP (0.37) SYKADORA3ADORA1USP7POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3781565-A1 2-METHYL-AZA-QUINAZOLINES Bayer Pharma Aktiengesellschaft (DE) 2021-02-24 EP disclosed
WO-2019201848-A1 2-METHYL-AZA-QUINAZOLINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2019-10-24 WO disclosed