SCHEMBL214953

SCHEMBL214953

CCCC1(N)N=C2N=CN=C2C(=O)N1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6536480 0.88 MPO (0.31)
SCHEMBL8046859 0.73
SCHEMBL6681436 0.73 ALDH1A1 (0.34)
SCHEMBL789177 0.71
SCHEMBL1377643 0.69
SCHEMBL6810692 0.63
Water SCHEMBL30522000 0.58 MPO (0.34)
SCHEMBL2523527 0.57 DHFR (0.34)
SCHEMBL4091048 0.53
SCHEMBL7535813 0.53 KDM4E (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2308 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12630827-B2 Antisense oligonucleotides targeting SCN2A for the treatment of SCN1A encephalopathies ROGCON, INC. (US) 2026-05-19 US claimed
EP-4705481-A2 CIRCULAR RNA COMPOSITIONS AND METHODS Orna Therapeutics, Inc. (US) 2026-03-11 EP claimed
US-20250257360-A1 OLIGONUCLEOTIDE INTERFERENCE TREATMENTS OF PROSTATE CANCER UNIV OKLAHOMA (US) 2025-08-14 US claimed
CN-113151261-B Antisense oligonucleotides as inhibitors of TGF-R signaling 神经视觉医药有限公司 2025-06-17 CN claimed
US-20250179503-A1 METHODS OF USING OLIGOMERIC COMPOUNDS TO TREAT SCN2A-RELATED DISORDERS PRAXIS PREC MEDICINES INC (US) 2025-06-05 US claimed
US-20250146073-A1 METHODS FOR THE TREATMENT OF SCN2A-RELATED DISORDERS PRAXIS PREC MEDICINES INC (US) 2025-05-08 US claimed
EP-4504945-A2 OLIGONUCLEOTIDE INTERFERENCE TREATMENTS OF PROSTATE CANCER The Board of Regents of the University of Oklahoma (US) 2025-02-12 EP claimed
EP-4499835-A2 METHODS OF USING OLIGOMERIC COMPOUNDS TO TREAT SCN2A-RELATED DISORDERS Praxis Precision Medicines, Inc. (US) 2025-02-05 EP claimed
EP-4473113-A2 METHODS FOR THE TREATMENT OF SCN2A-RELATED DISORDERS Praxis Precision Medicines, Inc. (US) 2024-12-11 EP claimed
US-12146139-B2 Oligonucleotide interference treatments of prostate cancer THE BOARD OF REGENTS OF THE UNIVERSITY OF OKLAHOMA (US) 2024-11-19 US claimed
WO-2016075339-A1 ANTISENSE-OLIGONUCLEOTIDES AS INHIBITORS OF TGF-R SIGNALING Neurovision Pharma GmbH (DE) 2016-05-19 WO claimed
EP-3020813-A1 Antisense-oligonucleotides as inhibitors of TGF-R signaling Neurovision Pharma GmbH (DE) 2016-05-18 EP claimed
US-9334495-B2 Minor groove binder (MGB)-oligonucleotide miRNA antagonists ELITECHGROUP B.V. (NL) 2016-05-10 US claimed
EP-2547769-A1 MINOR GROOVE BINDER (MGB)-OLIGONUCLEOTIDE MIRNA ANTAGONISTS Elitech Holding B.V. (NL) 2013-01-23 EP claimed
WO-2012099630-A1 COMPOSITIONS AND METHODS FOR TREATING OR PREVENTING A RETROVIRUS INFECTION UNIVERSITY OF ROCHESTER (US) 2012-07-26 WO claimed
US-20110172289-A1 MINOR GROOVE BINDER (MGB)-OLIGONUCLEOTIDE MIRNA ANTAGONISTS ELITECH HOLDING B.V. 2011-07-14 US claimed
WO-2011066312-A1 MINOR GROOVE BINDER (MGB)-OLIGONUCLEOTIDE MIRNA ANTAGONISTS ELITECH HOLDING B.V. (NL) 2011-06-03 WO claimed
US-7067497-B2 Modulation of telomere length by oligonucleotides having a G-core sequence ISIS PHARMACEUTICALS, INC. (US) 2006-06-27 US claimed
US-20040049022-A1 Composition &amp; methods for treatment and screening NYCE JONATHAN W (US) 2004-03-11 US claimed
WO-2004011613-A2 COMPOSITION &amp; METHODS FOR TREATMENT AND SCREENING EPIGENESIS PHARMACEUTICALS, INC. (US) 2004-02-05 WO claimed