SCHEMBL21496729

SCHEMBL21496729

O=C1CCC[C@H](C(F)(F)F)C1

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 2/20 0.36
NOS1 P29475 2/20 0.36
NOS2 P35228 2/20 0.36
MAPT P10636 1/20 0.35
THRB P10828 1/20 0.34
TRIM24 O15164 2/20 0.33
TRIM33 Q9UPN9 2/20 0.33
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24097335 1.00 NOS3 (0.36) NOS3NOS1NOS2MAPTTHRB
SCHEMBL1397564 1.00 NOS3 (0.36) NOS3NOS1NOS2MAPTTHRB
SCHEMBL29281259 0.86 NOS3 (0.39) NOS3NOS1NOS2
SCHEMBL28247829 0.82 TRIM24 (0.39) NOS3NOS1NOS2TRIM24TRIM33
SCHEMBL22792768 0.78 THRB (0.37) MAPTTHRB
SCHEMBL918723 0.77 THRB (0.38) MAPTTHRBTRIM24TRIM33ALDH1A1
SCHEMBL3973236 0.73 NOS3 (0.36) NOS3NOS1NOS2
SCHEMBL18535813 0.72 KEAP1 (0.45) ALDH1A1
SCHEMBL17247965 0.71 SLC2A1 (0.40) MAPTTHRBALDH1A1
SCHEMBL1711546 0.70 MAPT (0.34) NOS3NOS1NOS2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4110298-A1 HOT MELT EXTRUDED SOLID DISPERSIONS CONTAINING A BCL2 INHIBITOR Guangzhou Lupeng Pharmaceutical Company Ltd. (CN) 2023-01-04 EP disclosed
CN-113710812-A Process for producing (1R,3R) -3- (trifluoromethyl) cyclohexan-1-ol and intermediate thereof 株式会社API 2021-11-26 CN disclosed
EP-3784654-A1 ISOINDOLINES AS HDAC INHIBITORS Valo Early Discovery, Inc. (US) 2021-03-03 EP disclosed
WO-2020213731-A1 METHOD FOR PRODUCING (1R,3R)-3-(TRIFLUOROMETHYL)CYCLOHEXAN-1-OL AND INTERMEDIATE THEREOF 株式会社エーピーアイ コーポレーション 2020-10-22 WO disclosed
WO-2019204550-A1 ISOINDOLINES AS HDAC INHIBITORS FORMA THERAPEUTICS, INC. (US) 2019-10-24 WO disclosed