SCHEMBL21512972

SCHEMBL21512972

C=CS(=O)(=O)NC[C@H]1CCN(C(=O)/C(C)=C/C)C1

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
F10 P00742 14/20 0.37
ALDH1A1 P00352 4/20 0.37
LMNA P02545 1/20 0.37
POLB P06746 1/20 0.37
MAPT P10636 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21512973 0.90 F10 (0.38) F10ALDH1A1LMNAPOLBMAPT
SCHEMBL21512971 0.87 ALDH1A1 (0.39) F10ALDH1A1LMNAPOLBMAPT
SCHEMBL21496865 0.82 F10 (0.37) F10ALDH1A1LMNAPOLBCYP3A4
SCHEMBL21512153 0.77 ALDH1A1 (0.47) F10ALDH1A1CYP3A4CYP2D6CYP2C9
SCHEMBL21512799 0.77 ALDH1A1 (0.47) F10ALDH1A1CYP3A4CYP2D6CYP2C9
SCHEMBL21511818 0.76 ALDH1A1 (0.35) F10ALDH1A1LMNAPOLB
SCHEMBL21512168 0.76 ALDH1A1 (0.35) F10ALDH1A1LMNAPOLB
SCHEMBL21496890 0.75 ALDH1A1 (0.41) ALDH1A1LMNAPOLBMAPT
SCHEMBL21512968 0.74 ALDH1A1 (0.31) ALDH1A1
SCHEMBL21512966 0.72 DRD2 (0.34) ALDH1A1POLBCYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019204505-A2 K-RAS MODULATORS WITH A VINYL SULFONAMIDE MOIETY THERAS, INC. (US) 2019-10-24 WO disclosed