SCHEMBL21532910

SCHEMBL21532910

Cc1ncccc1CNN

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 4/20 0.49
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.43
CYP2C9 P11712 1/20 0.43
NAMPT P43490 1/20 0.43
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
NOS2 P35228 1/20 0.38
GABRA5 P31644 1/20 0.38
IL1B P01584 2/20 0.36
IDO1 P14902 1/20 0.35
DCPS Q96C86 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA2B P29275 1/20 0.35
JAK3 P52333 1/20 0.35
VCP P55072 1/20 0.35
PIK3CA P42336 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6047196 0.82 CYP2C9 (0.43) P2RX7CYP2C9NAMPTGABRA5
SCHEMBL21617369 0.80 P2RX7 (0.58) P2RX7ALDH1A1MAPTCYP2C9NAMPT
SCHEMBL17886855 0.78 CYP2C9 (0.42) P2RX7ALDH1A1GAACYP2C9NAMPT
SCHEMBL17888348 0.78 GAA (0.42) P2RX7GAACYP2C9NAMPTGABRA5
Hydrochloric Acid SCHEMBL31169752 0.78 CYP2C9 (0.42) P2RX7ALDH1A1CYP2C9NAMPT
SCHEMBL8550272 0.77 ADRA2C (0.46) P2RX7CYP2C9NAMPTGABRA5ADORA2A
SCHEMBL261850 0.77
SCHEMBL13401252 0.76 KDM1A (0.43) P2RX7ALDH1A1GAAMAPTIDO1
SCHEMBL13731868 0.76 CYP2C9 (0.59) P2RX7ALDH1A1GAAMAPTCYP2C9
Hydrochloric Acid SCHEMBL5010799 0.75 DPP4 (0.44) P2RX7CYP2C9NAMPTNOS3NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20190330181-A1 HEMOGLOBIN MODIFIER COMPOUNDS AND USES THEREOF SICHUAN HAISCO PHARMACEUTICAL CO., LTD. (CN) 2019-10-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190330181-A1 HEMOGLOBIN MODIFIER COMPOUNDS AND USES THEREOF HBB, HBG1, HBG2 P2RX7 4755/4885ALDH1A1 863/4885GAA 49/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.